HIV protease inhibitors

被引:12
作者
Molla, A
Japour, A
机构
关键词
D O I
10.1097/00001432-199712000-00015
中图分类号
R51 [传染病];
学科分类号
100401 ;
摘要
The past year has seen remarkable advances in the therapeutic options and strategies for the treatment of HIV infection. This review describes the recent clinical studies using protease inhibitors in combination therapy. Data on the emergence of protease inhibitor-conferring mutations, including drug resistance and the impact of further treatment options, are summarized.
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页码:491 / 495
页数:5
相关论文
共 29 条
[1]  
CAMERON DW, 1996, 11 INT C AIDS JUL 5
[2]  
CHAUVIN JP, 1996, INT C DRUG THER HIV
[3]   HIV POPULATION-DYNAMICS IN-VIVO - IMPLICATIONS FOR GENETIC-VARIATION, PATHOGENESIS, AND THERAPY [J].
COFFIN, JM .
SCIENCE, 1995, 267 (5197) :483-489
[4]   IN-VIVO EMERGENCE OF HIV-1 VARIANTS RESISTANT TO MULTIPLE PROTEASE INHIBITORS [J].
CONDRA, JH ;
SCHLEIF, WA ;
BLAHY, OM ;
GABRYELSKI, LJ ;
GRAHAM, DJ ;
QUINTERO, JC ;
RHODES, A ;
ROBBINS, HL ;
ROTH, E ;
SHIVAPRAKASH, M ;
TITUS, D ;
YANG, T ;
TEPPLER, H ;
SQUIRES, KE ;
DEUTSCH, PJ ;
EMINI, EA .
NATURE, 1995, 374 (6522) :569-571
[5]   A SHORT-TERM STUDY OF THE SAFETY, PHARMACOKINETICS, AND EFFICACY OF RITONAVIR, AN INHIBITOR OF HIV-1 PROTEASE [J].
DANNER, SA ;
CARR, A ;
LEONARD, JM ;
LEHMAN, LM ;
GUDIOL, F ;
GONZALES, J ;
RAVENTOS, A ;
RUBIO, R ;
BOUZA, E ;
PINTADO, V ;
AGUADO, AG ;
DELOMAS, JG ;
DELGADO, R ;
BORLEFFS, JCC ;
HSU, A ;
VALDES, JM ;
BOUCHER, CAB ;
COOPER, DA ;
GIMENO, C ;
CLOTET, B ;
TOR, J ;
FERRER, E ;
MARTINEZ, PL ;
MORENO, S ;
ZANCADA, G ;
ALCAMI, J ;
NORIEGA, AR ;
PULIDO, F ;
GLASSMAN, HN .
NEW ENGLAND JOURNAL OF MEDICINE, 1995, 333 (23) :1528-1533
[6]  
DANNER SA, 1996, INT C DRUG THER HIV
[7]  
DUBOUCK C, 1992, AIDS RES HUM RETROV, V8, P153
[8]   RESISTANCE OF HIV TYPE-1 TO PROTEINASE-INHIBITOR RO-31-8959 [J].
EBERLE, J ;
BECHOWSKY, B ;
ROSE, D ;
HAUSER, U ;
VONDERHELM, K ;
GURTLER, L ;
NITSCHKO, H .
AIDS RESEARCH AND HUMAN RETROVIRUSES, 1995, 11 (06) :671-676
[9]  
EMINI EA, 1997, INT WORKSH HIV DRUG
[10]   THE NOT-SO-GREAT ESCAPE [J].
ERICKSON, JW .
NATURE STRUCTURAL BIOLOGY, 1995, 2 (07) :523-529