Development of the Na+/H+ exchange inhibitor cariporide as a cardioprotective drug:: From the laboratory to the GUARDIAN trial

被引:18
作者
Scholz, W [1 ]
Jessel, A [1 ]
Albus, U [1 ]
机构
[1] Hoechst Marion Roussel, D-65926 Frankfurt, Germany
关键词
D O I
10.1023/A:1008998716063
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
[No abstract available]
引用
收藏
页码:61 / 69
页数:9
相关论文
共 27 条
[1]  
[Anonymous], 1988, LANCET, V2, P349
[2]  
ANTMAN EM, 1997, HEART DIS TXB CARDIO, P1184
[3]   Antiarrhythmic effects of cariporide, a novel Na+-H+ exchange inhibitor, on reperfusion ventricular arrhythmias in rat hearts [J].
Aye, NN ;
Xue, YX ;
Hashimoto, K .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1997, 339 (2-3) :121-127
[4]  
Bata I, 1997, CIRCULATION, V96, P769
[5]   Shattuck lecture - Cardiovascular medicine at the turn of the millennium: Triumphs, concerns, and opportunities [J].
Braunwald, E .
NEW ENGLAND JOURNAL OF MEDICINE, 1997, 337 (19) :1360-1369
[6]   USE OF A MONOCLONAL-ANTIBODY DIRECTED AGAINST THE PLATELET GLYCOPROTEIN IIB/IIIA RECEPTOR IN HIGH-RISK CORONARY ANGIOPLASTY [J].
CALIFF, RM ;
SHADOFF, N ;
VALETT, N ;
BATES, E ;
GALEANA, A ;
KNOPF, W ;
SHAFTEL, J ;
BENDER, MJ ;
AVERSANO, T ;
RAQUENO, J ;
GURBEL, P ;
COWFER, J ;
COHEN, M ;
CROSS, P ;
BITTL, J ;
EDDINGS, K ;
TAYLOR, M ;
DEROSA, K ;
HATTEL, L ;
COOPER, L ;
ESHELMAN, B ;
FINTEL, D ;
NIEMYSKI, P ;
KLEIN, L ;
KENNEDY, H ;
THORNTON, T ;
KEREIAKES, D ;
MARTIN, L ;
ANDERSON, L ;
HIGBY, N ;
ELLIS, S ;
BREZINA, K ;
GEORGE, B ;
CHAPEKIS, A ;
SMITH, D ;
ANWAR, A ;
GERBER, TL ;
PRITCHARD, GL ;
MYLER, R ;
SHAW, R ;
MURPHY, M ;
WARD, K ;
MADIGAN, NP ;
BLANKENSHIP, J ;
HALBERT, M ;
FLANAGAN, C ;
TANNENBAUM, M ;
POLICH, M ;
STEVENSON, C ;
TCHENG, J .
NEW ENGLAND JOURNAL OF MEDICINE, 1994, 330 (14) :956-961
[7]  
CEES JA, 1997, J MOL CELL CARDIOL, V29, pA28
[8]  
Drexler H, 1998, CIRCULATION, V98, P344
[9]   Prevention of ischemic rigor contracture during coronary occlusion by inhibition of Na+-H+ exchange [J].
GarciaDorado, D ;
Gonzalez, MA ;
Barrabes, JA ;
RuizMeana, M ;
Solares, J ;
Lidon, RM ;
Blanco, J ;
Puigfel, Y ;
Piper, HM ;
SolerSoler, J .
CARDIOVASCULAR RESEARCH, 1997, 35 (01) :80-89
[10]   NEW NA+-H+ EXCHANGE INHIBITOR HOE-694 IMPROVES POSTISCHEMIC FUNCTION AND HIGH-ENERGY PHOSPHATE RESYNTHESIS AND REDUCES CA2+ OVERLOAD IN ISOLATED-PERFUSED RABBIT HEART [J].
HENDRIKX, M ;
MUBAGWA, K ;
VERDONCK, F ;
OVERLOOP, K ;
VANHECKE, P ;
VANSTAPEL, F ;
VANLOMMEL, A ;
VERBEKEN, E ;
LAUWERYNS, J ;
FLAMENG, W .
CIRCULATION, 1994, 89 (06) :2787-2798