The Chemo- and Regioselectivity of the Cyclization of Thiosemicarbazides with Haloacetic Acids and their Derivatives

被引：5
作者：
Izmest'ev, Alexei N. [1 ]
Streltsov, Andrey A. [1 ]
Kravchenko, Angelina N. [1 ]
Gazieva, Galina A. [1 ]
机构：
[1] Russian Acad Sci, ND Zelinsky Inst Organ Chem, 47 Leninsky Ave, Moscow 119991, Russia
来源：
CHEMISTRY OF HETEROCYCLIC COMPOUNDS | 2022年 / 58卷 / 10期
关键词：
azines; azoles; thiazolidin-4-ones; thiosemicarbazides; cyclocondensation; regioselectivity; MICROWAVE-ASSISTED SYNTHESIS; BIOLOGICAL EVALUATION; THIAZOLIDINONE DERIVATIVES; INHIBITORS SYNTHESIS; FACILE SYNTHESIS; ANTIMICROBIAL ACTIVITIES; PHTHALAZINE DERIVATIVES; ANTICONVULSANT ACTIVITY; THIAZOLE DERIVATIVES; PYRIDINE-DERIVATIVES;
D O I：
10.1007/s10593-022-03117-3
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The effect of the structural features of the starting thiosemicarbazides as well as the cyclization reaction conditions on the chemo- and regioselectivity of the formation of heterocyclic systems is discussed.
引用
收藏
页码：483 / 492
页数：10
相关论文
共 191 条
[1]   Syntheses of new unsymmetrical and symmetrical diarylsulphides and diarylsulphones containing thiazolinyl and thiazolidinonyl moieties using 4,4′-diacetyidiphenylsulphide [J].
Abbady, MA ;
Abdel-Hafez, SH ;
Kandeel, MM ;
Abdel-Monem, MI .
MOLECULES, 2003, 8 (08) :622-641
[2]   Synthesis and Structure-Activity Relationship Study of Novel Pyrazolylthiazoles as Potential Anti-Breast Cancer Agents [J].
Abbas, Eman M. H. ;
Dawood, Dina H. ;
Farghaly, Thoraya A. ;
El-hag, Fatma A. ;
Ali, Mamdouh M. .
JOURNAL OF HETEROCYCLIC CHEMISTRY, 2017, 54 (03) :1974-1982
[3]   Synthesis of fused 1,2,4-triazines as potential antimicrobial and antitumor agents [J].
Abd El-Moneim, Mohamed ;
Hasanen, J. A. ;
El-Deen, I. M. ;
Abd El-Fattah, W. .
RESEARCH ON CHEMICAL INTERMEDIATES, 2015, 41 (06) :3543-3561
[4]   A facile synthesis of some novel thiazoles, arylazothiazoles, and pyrazole linked to thiazolyl coumarin as antibacterial agents [J].
Abdel-Aziem, Anhar ;
Baaiu, Basma Saad ;
Elbazzar, Awad Wanis ;
Elabbar, Fakhri .
SYNTHETIC COMMUNICATIONS, 2020, 50 (16) :2522-2530
[5]   Synthesis and Biological Studies of Some New Thiazoles, Hydrazones and Azine Derivatives Based on 3,5-Diphenylcyclohex-2-en-1-one [J].
Abdel-Galil, Ebrahim ;
Girges, Margret M. ;
Said, Gehad E. .
CHEMISTRYSELECT, 2020, 5 (10) :3075-3079
[6]  
Abdel-Rahman, 2007, EGYPT J CHEM, V50, P771
[7]  
Abdel-Rahman A. H., 2013, Der Pharm. Chem, V5, P210
[8]  
Abdel-Rahman RM., 1992, ASIAN J CHEM, V4, P534
[9]  
Abdel-Samii Z.K., 2017, World J. Pharm. Res., V6, P1450, DOI [10.20959/wjpr20172-7874, DOI 10.20959/WJPR20172-7874]
[10]   Synthesis of New 7-Oxycoumarin Derivatives As Potent and Selective Monoamine Oxidase A Inhibitors [J].
Abdelhafez, Omaima M. ;
Amin, Kamelia M. ;
Ali, Hamed I. ;
Abdalla, Mohamed M. ;
Batran, Rasha Z. .
JOURNAL OF MEDICINAL CHEMISTRY, 2012, 55 (23) :10424-10436
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