The antiarrhythmic drug mexiletine blocks HERG potassium channels

被引:0
|
作者
Qu, YS [1 ]
Qian, YX [1 ]
McGivern, J [1 ]
机构
[1] Amgen Inc, Thousand Oaks, CA 91320 USA
关键词
D O I
暂无
中图分类号
Q6 [生物物理学];
学科分类号
071011 ;
摘要
2860
引用
收藏
页码:585A / 585A
页数:1
相关论文
共 50 条
  • [1] Antiarrhythmic drug carvedilol inhibits HERG potassium channels
    Karle, CA
    Kreye, VAW
    Thomas, D
    Röckl, K
    Kathöfer, S
    Zhang, W
    Kiehn, J
    CARDIOVASCULAR RESEARCH, 2001, 49 (02) : 361 - 370
  • [2] Cocaine blocks HERG potassium channels
    Zhang, ST
    Zhou, ZF
    Chen, YM
    Gong, QM
    Ruoho, AE
    January, CT
    CIRCULATION, 1999, 100 (18) : 424 - 424
  • [3] Inhibitory effects of the class III antiarrhythmic drug amiodarone on cloned HERG potassium channels
    J. Kiehn
    Dierk Thomas
    Christoph A. Karle
    Wolfgang Schöls
    Wolfgang Kübler
    Naunyn-Schmiedeberg's Archives of Pharmacology, 1999, 359 : 212 - 219
  • [4] Inhibitory effects of the class III antiarrhythmic drug amiodarone on cloned HERG potassium channels
    Kiehn, J
    Thomas, D
    Karle, CA
    Schöls, W
    Kübler, W
    NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1999, 359 (03) : 212 - 219
  • [5] Inhibition of hERG potassium channel by the antiarrhythmic agent mexiletine and its metabolite m-hydroxymexiletine
    Gualdani, Roberta
    Tadini-Buoninsegni, Francesco
    Roselli, Mariagrazia
    Defrenza, Ivana
    Contino, Marialessandra
    Colabufo, Nicola Antonio
    Lentini, Giovanni
    PHARMACOLOGY RESEARCH & PERSPECTIVES, 2015, 3 (05):
  • [6] Blocking effects of the antiarrhythmic drug propafenone on the HERG potassium channel
    Mergenthaler, J
    Haverkamp, W
    Hüttenhofer, A
    Skryabin, BV
    Musshoff, U
    Borggrefe, M
    Speckmann, EJ
    Breithardt, G
    Madeja, M
    NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 2001, 363 (04) : 472 - 480
  • [7] Blocking effects of the antiarrhythmic drug propafenone on the HERG potassium channel
    Jörg Mergenthaler
    Wilhelm Haverkamp
    Alexander Hüttenhofer
    Boris V. Skryabin
    Ulrich Mußhoff
    Martin Borggrefe
    Erwin-Josef Speckmann
    Günter Breithardt
    Michael Madeja
    Naunyn-Schmiedeberg's Archives of Pharmacology, 2001, 363 : 472 - 480
  • [8] Bertosamil blocks HERG potassium channels in their open and inactivated states
    Zitron, E
    Karle, CA
    Wendt-Nordahl, G
    Kathöfer, S
    Zhang, W
    Thomas, D
    Weretka, S
    Kiehn, J
    BRITISH JOURNAL OF PHARMACOLOGY, 2002, 137 (02) : 221 - 228
  • [9] Aconitine blocks HERG and Kv1.5 potassium channels
    Li, Yifu
    Tu, Danna
    Xiao, Hua
    Du, Yimei
    Zou, Anruo
    Liao, Yuhua
    Dong, Shaohong
    JOURNAL OF ETHNOPHARMACOLOGY, 2010, 131 (01) : 187 - 195
  • [10] Class Ia anti-arrhythmic drug ajmaline blocks HERG potassium channels: mode of action
    Claudia Kiesecker
    Edgar Zitron
    Sonja Lück
    Ramona Bloehs
    Eberhard P. Scholz
    Sven Kathöfer
    Dierk Thomas
    Volker A. W. Kreye
    Hugo A. Katus
    Wolfgang Schoels
    Christoph A. Karle
    Johann Kiehn
    Naunyn-Schmiedeberg's Archives of Pharmacology, 2004, 370 : 423 - 435