Efficient one-pot three-component synthesis of 7-oxo-1,7,8,8a-tetrahydroimidazo[1,2-α]pyrimidines

被引：20

作者：

Adib, M ^{[1
]}

Mollahosseini, M

Yavari, H

Sayahi, MH

Bijanzadeh, HR

机构：

[1] Univ Tehran, Fac Sci, Dept Chem, Tehran, Iran

[2] Univ Tarbiat Modarres, Dept Chem, Tehran, Iran

来源：

SYNLETT | 2004年 / 06期

关键词：

isocyanates; cyclizations; heterocycles; imidazoles; alkynes;

D O I：

10.1055/s-2004-820056

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

1-Methyl imidazole reacts smoothly with dialkyl acetylenedicarboxylates in the presence of isocyanates to produce dialkyl 1-methyl-7-oxo-1,7,8,8a-tetrahydroimidazo[1,2-a]pyrimidine-5,6-dicarboxylates in excellent yields.

引用

页码：1086 / 1088

页数：3

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