共 50 条
- [1] From DNA-Encoded Library Screening to AM-9747: An MTA-Cooperative PRMT5 Inhibitor with Potent Oral In Vivo EfficacyJOURNAL OF MEDICINAL CHEMISTRY, 2025, 68 (06) : 6534 - 6557Sarvary, Ian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkVestergaard, Mikkel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkMoretti, Loris论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkAndersson, Jan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkCadahia, Jorge Peiro论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkCowland, Sanne论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkFlagstad, Thomas论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkFranch, Thomas论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkGouliaev, Alex论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkHusemoen, Gitte论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkJacso, Tomas论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkKronborg, Titi论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkKuropatnicka, Aleksandra论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkNadali, Anna论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkMadsen, Mads论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkNielsen, Soren论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkPii, David论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkRyborg, Soren论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkSoede, Camillia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkAllen, Jennifer R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkBourbeau, Matthew论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkLi, Kexue论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkLiu, Qingyian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkLo, Mei-Chu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, South San Francisco, CA 94080 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkMadoux, Franck论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkMardirossian, Narbe论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkMoriguchi, Jodi论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkNgo, Rachel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, South San Francisco, CA 94080 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkPeng, Chi-Chi论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, South San Francisco, CA 94080 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkPettus, Liping论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkTamayo, Nuria论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkWang, Paul论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkKapoor, Rajiv论文数: 0 引用数: 0 h-index: 0机构: Amgen Res, Syngene Amgen Res & Dev Ctr, Bangalore 560099, India Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkBelmontes, Brian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkCaenepeel, Sean论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkHughes, Paul论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkLiu, Siyuan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkSlemmons, Katherine K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkYang, Yajing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkXie, Fang论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, South San Francisco, CA 94080 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkGhimire-Rijal, Sudipa论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkMukund, Susmith论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, DK-2100 Copenhagen, DenmarkGlad, Sanne论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark Amgen Inc, Amgen Res, DK-2100 Copenhagen, Denmark
- [2] iscovery and characterization of an MTA-cooperative and brain-penetrant PRMT5 inhibitorMOLECULAR CANCER THERAPEUTICS, 2023, 22 (12)Pan, Welling论文数: 0 引用数: 0 h-index: 0Wang, Hui论文数: 0 引用数: 0 h-index: 0Qi, Fangfei论文数: 0 引用数: 0 h-index: 0Deng, Haibing论文数: 0 引用数: 0 h-index: 0Yang, Fei论文数: 0 引用数: 0 h-index: 0Yu, Hongping论文数: 0 引用数: 0 h-index: 0Xu, Yao-Chang论文数: 0 引用数: 0 h-index: 0Chen, Zhui论文数: 0 引用数: 0 h-index: 0Ying, Haiyan论文数: 0 引用数: 0 h-index: 0
- [3] Preclinical characterization of ABSK131, a potential best-in-class MTA-cooperative PRMT5 inhibitorEUROPEAN JOURNAL OF CANCER, 2024, 211 : S17 - S18Pan, W.论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Biol, Shanghai, Peoples R China Abbisko Therapeut, Biol, Shanghai, Peoples R ChinaWang, H.论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Biol, Shanghai, Peoples R China Abbisko Therapeut, Biol, Shanghai, Peoples R ChinaQi, F.论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Biol, Shanghai, Peoples R China Abbisko Therapeut, Biol, Shanghai, Peoples R ChinaDeng, H.论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Chem, Shanghai, Peoples R China Abbisko Therapeut, Biol, Shanghai, Peoples R ChinaYu, H.论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Chem, Shanghai, Peoples R China Abbisko Therapeut, Biol, Shanghai, Peoples R ChinaXu, Y. C.论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Chem, Shanghai, Peoples R China Abbisko Therapeut, Biol, Shanghai, Peoples R ChinaChen, Z.论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Biol, Shanghai, Peoples R China Abbisko Therapeut, Biol, Shanghai, Peoples R ChinaYing, H.论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Biol, Shanghai, Peoples R China Abbisko Therapeut, Biol, Shanghai, Peoples R China
- [4] Discovery of AMG 193, an MTA-Cooperative PRMT5 Inhibitor for the Treatment of MTAP-Deleted CancersJOURNAL OF MEDICINAL CHEMISTRY, 2025,Pettus, Liping H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USABourbeau, Matthew论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USATamayo, Nuria A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAAmegadzie, Albert论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USABeylkin, Diane论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USABooker, Shon K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAButler, John论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAFrohn, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAKaller, Matthew R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAKohn, Todd论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USALanman, Brian A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USALi, Kexue论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USALiu, Qingyian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAMa, Vu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAMedina, Jose论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAMinatti, Ana E.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USALopez, Patricia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAManoni, Francesco论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAPickrell, Alex论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAWeires, Nicholas论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAAndersson, Jan论文数: 0 引用数: 0 h-index: 0机构: Amgen Res Copenhagen, Small Mol Therapeut Discovery, DK-2100 Copenhagen, Denmark Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USACowland, Sanne论文数: 0 引用数: 0 h-index: 0机构: Amgen Res Copenhagen, Small Mol Therapeut Discovery, DK-2100 Copenhagen, Denmark Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAGlad, Sanne论文数: 0 引用数: 0 h-index: 0机构: Amgen Res Copenhagen, Small Mol Therapeut Discovery, DK-2100 Copenhagen, Denmark Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USASarvary, Ian论文数: 0 引用数: 0 h-index: 0机构: Amgen Res Copenhagen, Small Mol Therapeut Discovery, DK-2100 Copenhagen, Denmark Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAVestergaard, Mikkel论文数: 0 引用数: 0 h-index: 0机构: Amgen Res Copenhagen, Small Mol Therapeut Discovery, DK-2100 Copenhagen, Denmark Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USALi, Weikun论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Drug Prod Technol, Proc Dev, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAGhimire-Rijal, Sudipa论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAMardirossian, Narbe论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAMukund, Susmith论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAChen, Qing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USALo, Mei-Chu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, South San Francisco, CA 94080 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USANgo, Rachel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, South San Francisco, CA 94080 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAKhetan, Jawahar论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAMadoux, Franck论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USASanders, Christiana论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USASharma, Pooja论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAWang, Paul论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USABruenner, Bernd论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, TS&BA Bioanalyt Sci, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAMccloud, Stuart论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, TS&BA Bioanalyt Sci, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAPonce, Manuel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Pharmacokinet & Drug Metab, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USASoto, Marcus论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Pharmacokinet & Drug Metab, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAWahlstrom, Jan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pharmacokinet & Drug Metab, Amgen Res, San Francisco, CA 94080 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAXie, Fang论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pharmacokinet & Drug Metab, Amgen Res, San Francisco, CA 94080 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAYang, Yajing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USALiu, Siyuan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USATan, Hong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USAPolicheni, Antonia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USACaenepeel, Sean论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USASlemmons, Katherine K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USABelmontes, Brian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Small Mol Therapeut Discovery, Amgen Res, Thousand Oaks, CA 91320 USA
- [5] The discovery and preclinical characterization of AMG 193, a first-in-class MTA-cooperative PRMT5 inhibitor with broad activity against MTAP-null cancersMOLECULAR CANCER THERAPEUTICS, 2023, 22 (12)Bojko-Matuszek, Agnieszka论文数: 0 引用数: 0 h-index: 0Kolakowski, Damian论文数: 0 引用数: 0 h-index: 0Bojko, Magdalena论文数: 0 引用数: 0 h-index: 0Sowinska, Aleksandra论文数: 0 引用数: 0 h-index: 0Mitula, Filip论文数: 0 引用数: 0 h-index: 0Lacek, Krzysztof论文数: 0 引用数: 0 h-index: 0Popiel, Delfina论文数: 0 引用数: 0 h-index: 0Kwiatkowski, Sebastian论文数: 0 引用数: 0 h-index: 0Kornatowski, Tomasz论文数: 0 引用数: 0 h-index: 0Kliszcz, Beata论文数: 0 引用数: 0 h-index: 0Jablonska, Anna论文数: 0 引用数: 0 h-index: 0Flis, Krzysztof论文数: 0 引用数: 0 h-index: 0Wiernicki, Bartosz论文数: 0 引用数: 0 h-index: 0Wieczorek, Maciej论文数: 0 引用数: 0 h-index: 0Pieczykolan, Jerzy论文数: 0 引用数: 0 h-index: 0Abramczyk, Olga论文数: 0 引用数: 0 h-index: 0
- [6] The discovery and preclinical characterization of the SAM-competitive PRMT5 inhibitor UCT-000445CANCER RESEARCH, 2023, 83 (07)McDermott, Martina S.论文数: 0 引用数: 0 h-index: 0O'Brien, Neil A.论文数: 0 引用数: 0 h-index: 0O'Boyle, Brendan论文数: 0 引用数: 0 h-index: 0Bartberger, Michael论文数: 0 引用数: 0 h-index: 0Loson, Oliver C.论文数: 0 引用数: 0 h-index: 0Chau, Kevin论文数: 0 引用数: 0 h-index: 0Schwab, Ella论文数: 0 引用数: 0 h-index: 0Hong, Jenny论文数: 0 引用数: 0 h-index: 0Zhou, Jiaying论文数: 0 引用数: 0 h-index: 0Hu, Chuhong论文数: 0 引用数: 0 h-index: 0Luo, Tong论文数: 0 引用数: 0 h-index: 0Ayala, Raul论文数: 0 引用数: 0 h-index: 0Glasby, John论文数: 0 引用数: 0 h-index: 0Stoltz, Brian M.论文数: 0 引用数: 0 h-index: 0Slamon, Dennis J.论文数: 0 引用数: 0 h-index: 0
- [7] A review of the known MTA-cooperative PRMT5 inhibitorsRSC Advances, 2024, 14 (53) : 39653 - 39691Hu, Mei论文数: 0 引用数: 0 h-index: 0机构: Department of Pharmaceutical Sciences, School of Pharmacy, Southwest Medical University, 1-1 Xiangling Road, Sichuan, Luzhou,646000, China Department of Pharmaceutical Sciences, School of Pharmacy, Southwest Medical University, 1-1 Xiangling Road, Sichuan, Luzhou,646000, ChinaChen, Xiang论文数: 0 引用数: 0 h-index: 0机构: Department of Pharmaceutical Sciences, School of Pharmacy, Southwest Medical University, 1-1 Xiangling Road, Sichuan, Luzhou,646000, China Department of Pharmaceutical Sciences, School of Pharmacy, Southwest Medical University, 1-1 Xiangling Road, Sichuan, Luzhou,646000, China
- [8] Discovery of highly selective novel MTA-cooperative PRMT5 inhibitors for the treatment of cancersCANCER RESEARCH, 2024, 84 (06)Wu, Wen-Lian论文数: 0 引用数: 0 h-index: 0Hu, Taishan论文数: 0 引用数: 0 h-index: 0Deng, Zhilin论文数: 0 引用数: 0 h-index: 0Li, Honghai论文数: 0 引用数: 0 h-index: 0Shen, Quanrong论文数: 0 引用数: 0 h-index: 0Zhang, Lei论文数: 0 引用数: 0 h-index: 0Ma, Xiaochu论文数: 0 引用数: 0 h-index: 0Sun, Peihua论文数: 0 引用数: 0 h-index: 0Cheng, Cindy论文数: 0 引用数: 0 h-index: 0Liu, Fang论文数: 0 引用数: 0 h-index: 0Chen, Xin论文数: 0 引用数: 0 h-index: 0Hua, Ye论文数: 0 引用数: 0 h-index: 0Huang, Bryan论文数: 0 引用数: 0 h-index: 0
- [9] TNG908, a brain-penetrant MTA-cooperative PRMT5 inhibitor, is efficacious in preclinical glioblastoma modelsCANCER RESEARCH, 2023, 83 (07)Zhang, Minjie论文数: 0 引用数: 0 h-index: 0Tsai, Alice论文数: 0 引用数: 0 h-index: 0Cottrell, Kevin M.论文数: 0 引用数: 0 h-index: 0Haines, Brian B.论文数: 0 引用数: 0 h-index: 0Wilker, Erik论文数: 0 引用数: 0 h-index: 0DiBenedetto, Heather论文数: 0 引用数: 0 h-index: 0Weitzman, Ron论文数: 0 引用数: 0 h-index: 0Huang, Alan论文数: 0 引用数: 0 h-index: 0Davis, Charles B.论文数: 0 引用数: 0 h-index: 0Maxwell, John P.论文数: 0 引用数: 0 h-index: 0Briggs, Kimberly J.论文数: 0 引用数: 0 h-index: 0
- [10] Discovery and In Vivo Efficacy of AZ-PRMT5i-1, a Novel PRMT5 Inhibitor with High MTA CooperativityJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (16) : 13604 - 13638Smith, James M.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandBarlaam, Bernard论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandBeattie, David论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandBradshaw, Lauren论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandChan, Ho Man论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Waltham, MA 02451 USA AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandChiarparin, Elisabetta论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandCollingwood, Olga论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandCooke, Sophie L.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandCronin, Anna论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandCumming, Iain论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandDean, Emma论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandDebreczeni, Judit E.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, Englanddel Barco Barrantes, Ivan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandDiene, Coura论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandGianni, Davide论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandGuerot, Carine论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandGuo, Xiaoxiao论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandGuven, Sinem论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandHayhow, Thomas G.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandHong, Ted论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Waltham, MA 02451 USA AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandKemmitt, Paul D.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandLamont, Gillian M.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandLamont, Scott论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandLynch, James T.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandMcWilliams, Lisa论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandMoore, Shaun论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandRaubo, Piotr论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandRobb, Graeme R.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandRobinson, James论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandScott, James S.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandSrinivasan, Bharath论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandSteward, Oliver论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandStubbs, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandSyson, Karl论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandTan, Lixiang论文数: 0 引用数: 0 h-index: 0机构: Pharmaron Beijing Co Ltd, Beijing 100176, Peoples R China AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandTurner, Oliver论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandUnderwood, Elizabeth论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandUrosevic, Jelena论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandVazquez-Chantada, Mercedes论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandWhittaker, Amy L.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci Biopharmaceut R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandWilson, David M.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, EnglandWinter-Holt, Jon J.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England AstraZeneca, Res & Early Dev Oncol R&D, Cambridge CB2 0AA, England