The first synthesis of a 15-membered macrocycle. Model of ring I of kistamycin

被引：8

作者：

Roussi, G

Zamora, EG

Carbonnelle, AC

Beugelmans, R

机构：

[1] Inst. Chim. Substances Naturelles, CNRS, 91198, Gif-sur-Yvette

来源：

TETRAHEDRON LETTERS | 1997年 / 38卷 / 25期

关键词：

D O I：

10.1016/S0040-4039(97)00941-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The intramolecular SNAr reaction of a linear peptid precursor, whose termini carry respectively an ortho fluoro-nitro group and a phenol function, gives the 15-membered ring compound in good yield, under mild conditions. (C) 1997 Published by Elsevier Science Ltd.

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页码：4405 / 4406

页数：2

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