Utility of N′-((2-chloroquinolin-3-yl)methylene)-2-cyanoacetohydrazide as a Source of Biologically Active Novel Heterocycles

被引:4
|
作者
Elsayed, Galal A. [1 ]
Omara, Samir A. [1 ]
Kamel, Rabaa M. [1 ]
机构
[1] Ain Shams Univ, Fac Sci, Dept Chem, Cairo 11566, Egypt
关键词
SUBSTITUTED QUINOLINES; ACRIDONE ALKALOIDS; ANTICANCER DRUGS; DERIVATIVES; AGENTS; QUINAZOLINE; ANTAGONISTS; ANALOGS; DESIGN; ALKYL;
D O I
10.1002/jhet.2965
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
The title compound is used as a precursor in synthesis of differently sized heterocyclic systems bearing quinoline moeity. Investigation of antimicrobial activity of the new products was evaluated using agar well diffusion method against six reference microbial isolates. Most of the new compounds are potent as antimicrobial agents.
引用
收藏
页码:3427 / 3433
页数:7
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