Advance in C-H Arylation of Indoles

被引：11

作者：

Luo, Junfei ^{[1
]}

Xu, Xing ^{[1
]}

Zheng, Junliang ^{[1
]}

机构：

[1] Ningbo Univ, Sch Mat Sci & Chem Engn, Ningbo 315211, Zhejiang, Peoples R China

来源：

CHINESE JOURNAL OF ORGANIC CHEMISTRY | 2018年 / 38卷 / 02期

关键词：

transition-metal catalysis; C-H bond activation; indoles; arylation; DIRECT C-2 ARYLATION; CATALYZED DIRECT ARYLATION; 2ND TOTAL-SYNTHESIS; ROOM-TEMPERATURE; BOND ARYLATION; SELECTIVE ARYLATION; DIRECT C2-ARYLATION; N-PIVALOYLINDOLES; FREE (NH)-INDOLES; METAL-FREE;

D O I：

10.6023/cjoc201707031

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The indoles motifs are widely found in the nature. One of the efficient strategy to access the indole derivatives is through the direct C-H functionalization of indole framework itself under transition-metal catalysis. Herein, the research advances on the transition-metal-catalyzed C-H arylation of indoles are reviewed.

引用

页码：363 / 377

页数：15

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