Synthesis and Insecticidal Activities of Novel Analogues of Flubendiamide Containing a Hexafluoroisopropanol Moiety

被引:3
作者
Wu Mingxi [1 ]
Zhao Wenwen [1 ]
Jin Guanyi [1 ]
Huang Qingchun [1 ]
Cao Song [1 ]
机构
[1] E China Univ Sci & Technol, Sch Pharm, Shanghai Key Lab Chem Biol, Shanghai 200237, Peoples R China
基金
国家高技术研究发展计划(863计划); 中国国家自然科学基金;
关键词
hexafluoroisopropanol moiety; flubendiamide; synthesis; insecticidal activities; DESIGN; FLUORINE; ACID; DERIVATIVES; RECEPTOR;
D O I
10.1002/cjoc.201200215
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
Ten novel analogues of flubendiamide containing a hexafluoroisopropanol moiety were designed and synthesized. Their insecticidal activities against armyworm (Pseudaletia separata Walker) were examined and compared with the commercial product flubendiamide. Compound 7b showed nearly the same insecticidal activity as flubendiamide against armyworm.
引用
收藏
页码:1310 / 1314
页数:5
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