Lithocholic acid analogues, new and potent α-2,3-sialyltransferase inhibitors

被引：59

作者：

Chang, KH

Lee, L

Chen, J

Li, WS ^{[1
]}

机构：

[1] Acad Sinica, Inst Chem, Taipei 115, Taiwan

[2] Natl Taiwan Normal Univ, Dept Chem, Taipei 116, Taiwan

来源：

CHEMICAL COMMUNICATIONS | 2006年 / 06期

关键词：

D O I：

10.1039/b514915k

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A new type of noncompetitive alpha-2,3-sialyltransferase inhibitor has been synthesized; we report the discovery, preparation and inhibitory activity of sixteen lithocholic acid analogues.

引用

页码：629 / 631

页数：3

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