共 47 条
Sulfamic acid: an efficient, cost-effective and recyclable catalyst for the synthesis of triazole[1,2-a]indazole-trione derivatives
被引:21
作者:

Kidwai, Mazaahir
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机构:
Univ Delhi, Dept Chem, Green Chem Res Lab, Delhi 110007, India Univ Delhi, Dept Chem, Green Chem Res Lab, Delhi 110007, India

Chauhan, Ritika
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机构:
Univ Delhi, Dept Chem, Green Chem Res Lab, Delhi 110007, India Univ Delhi, Dept Chem, Green Chem Res Lab, Delhi 110007, India
机构:
[1] Univ Delhi, Dept Chem, Green Chem Res Lab, Delhi 110007, India
来源:
关键词:
MULTICOMPONENT REACTIONS;
ONE-POT;
ORGANIC-REACTIONS;
URAZOLE;
INHIBITORS;
D O I:
10.1039/c2ra20662e
中图分类号:
O6 [化学];
学科分类号:
0703 ;
摘要:
Sulfamic acid (SA) is successfully utilized as a green, cost-effective and reusable catalyst for the synthesis of triazole[1,2-a]indazole-trione derivatives involving the one-pot, three-component condensation of urazole, aldehydes and cyclic beta-diketones in high yields in water as a sole solvent. The salient features of this new methodology are cheaper process, easy availability of the catalyst, mild conditions, versatility, and the catalyst could be recycled easily without affecting the catalytic activity.
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页码:7660 / 7665
页数:6
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共 47 条
[1]
Asymmetric synthesis of (3S,4R,5R)-4,5-dihydroxy-3-methyl-2,3,4,5-tetrahydropyridazine:: a formal synthesis of 1-azagulofagomine analogues
[J].
Arroyo, Y
;
Rodríguez, JF
;
Santos, M
;
Tejedor, MAS
;
Vaca, I
;
Ruano, JLG
.
TETRAHEDRON-ASYMMETRY,
2004, 15 (06)
:1059-1063

Arroyo, Y
论文数: 0 引用数: 0
h-index: 0
机构: Univ Valladolid, Dept Organ Chem, E-47011 Valladolid, Spain

Rodríguez, JF
论文数: 0 引用数: 0
h-index: 0
机构: Univ Valladolid, Dept Organ Chem, E-47011 Valladolid, Spain

Santos, M
论文数: 0 引用数: 0
h-index: 0
机构: Univ Valladolid, Dept Organ Chem, E-47011 Valladolid, Spain

Tejedor, MAS
论文数: 0 引用数: 0
h-index: 0
机构: Univ Valladolid, Dept Organ Chem, E-47011 Valladolid, Spain

Vaca, I
论文数: 0 引用数: 0
h-index: 0
机构: Univ Valladolid, Dept Organ Chem, E-47011 Valladolid, Spain

Ruano, JLG
论文数: 0 引用数: 0
h-index: 0
机构: Univ Valladolid, Dept Organ Chem, E-47011 Valladolid, Spain
[2]
Synthesis of novel lactam derivatives and their evaluation as ligands for the dopamine receptors, leading to a D4-selective ligand
[J].
Awadallah, Fadi M.
;
Mueller, Franziska
;
Lehmann, Jochen
;
Abadi, Ashraf H.
.
BIOORGANIC & MEDICINAL CHEMISTRY,
2007, 15 (17)
:5811-5818

Awadallah, Fadi M.
论文数: 0 引用数: 0
h-index: 0
机构: German Univ Cairo, Fac Pharm & Biotechnol, Dept Pharmaceut Chem, Cairo, Egypt

Mueller, Franziska
论文数: 0 引用数: 0
h-index: 0
机构: German Univ Cairo, Fac Pharm & Biotechnol, Dept Pharmaceut Chem, Cairo, Egypt

Lehmann, Jochen
论文数: 0 引用数: 0
h-index: 0
机构: German Univ Cairo, Fac Pharm & Biotechnol, Dept Pharmaceut Chem, Cairo, Egypt

Abadi, Ashraf H.
论文数: 0 引用数: 0
h-index: 0
机构:
German Univ Cairo, Fac Pharm & Biotechnol, Dept Pharmaceut Chem, Cairo, Egypt German Univ Cairo, Fac Pharm & Biotechnol, Dept Pharmaceut Chem, Cairo, Egypt
[3]
Rapid synthesis of VX-745: p38 MAP kinase inhibition in Werner syndrome cells
[J].
Bagley, Mark C.
;
Davis, Terence
;
Dix, Matthew C.
;
Rokicki, Michal J.
;
Kipling, David
.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
2007, 17 (18)
:5107-5110

Bagley, Mark C.
论文数: 0 引用数: 0
h-index: 0
机构: Univ Cardiff Wales, Sch Chem, Cardiff CF10 3AT, Wales

Davis, Terence
论文数: 0 引用数: 0
h-index: 0
机构: Univ Cardiff Wales, Sch Chem, Cardiff CF10 3AT, Wales

Dix, Matthew C.
论文数: 0 引用数: 0
h-index: 0
机构: Univ Cardiff Wales, Sch Chem, Cardiff CF10 3AT, Wales

Rokicki, Michal J.
论文数: 0 引用数: 0
h-index: 0
机构: Univ Cardiff Wales, Sch Chem, Cardiff CF10 3AT, Wales

Kipling, David
论文数: 0 引用数: 0
h-index: 0
机构: Univ Cardiff Wales, Sch Chem, Cardiff CF10 3AT, Wales
[4]
A novel three-component method for the synthesis of triazolo[1,2-a]indazole-triones
[J].
Bazgir, Ayoob
;
Seyyedhamzeh, Mozhdeh
;
Yasaei, Zahra
;
Mirzaei, Peiman
.
TETRAHEDRON LETTERS,
2007, 48 (50)
:8790-8794

Bazgir, Ayoob
论文数: 0 引用数: 0
h-index: 0
机构:
Shaheed Beheshti Univ Med Sci, Dept Chem, Tehran, Iran Shaheed Beheshti Univ Med Sci, Dept Chem, Tehran, Iran

Seyyedhamzeh, Mozhdeh
论文数: 0 引用数: 0
h-index: 0
机构:
Shaheed Beheshti Univ Med Sci, Dept Chem, Tehran, Iran Shaheed Beheshti Univ Med Sci, Dept Chem, Tehran, Iran

Yasaei, Zahra
论文数: 0 引用数: 0
h-index: 0
机构:
Shaheed Beheshti Univ Med Sci, Dept Chem, Tehran, Iran Shaheed Beheshti Univ Med Sci, Dept Chem, Tehran, Iran

Mirzaei, Peiman
论文数: 0 引用数: 0
h-index: 0
机构:
Shaheed Beheshti Univ Med Sci, Dept Chem, Tehran, Iran Shaheed Beheshti Univ Med Sci, Dept Chem, Tehran, Iran
[5]
High-throughput synthesis and optimization of thrombin inhibitors via urazole α-addition and Michael addition
[J].
Boatman, PD
;
Urban, J
;
Nguyen, M
;
Qabar, M
;
Kahn, M
.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
2003, 13 (08)
:1445-1449

Boatman, PD
论文数: 0 引用数: 0
h-index: 0
机构: Molecumetics, Bellevue, WA 98005 USA

Urban, J
论文数: 0 引用数: 0
h-index: 0
机构: Molecumetics, Bellevue, WA 98005 USA

Nguyen, M
论文数: 0 引用数: 0
h-index: 0
机构: Molecumetics, Bellevue, WA 98005 USA

Qabar, M
论文数: 0 引用数: 0
h-index: 0
机构: Molecumetics, Bellevue, WA 98005 USA

Kahn, M
论文数: 0 引用数: 0
h-index: 0
机构: Molecumetics, Bellevue, WA 98005 USA
[6]
Determining the geometries of transition states by use of antihydrophohic additives in water
[J].
Breslow, R
.
ACCOUNTS OF CHEMICAL RESEARCH,
2004, 37 (07)
:471-478

Breslow, R
论文数: 0 引用数: 0
h-index: 0
机构:
Columbia Univ, Dept Chem, New York, NY 10027 USA Columbia Univ, Dept Chem, New York, NY 10027 USA
[7]
HYDROPHOBIC EFFECTS ON SIMPLE ORGANIC-REACTIONS IN WATER
[J].
BRESLOW, R
.
ACCOUNTS OF CHEMICAL RESEARCH,
1991, 24 (06)
:159-164

BRESLOW, R
论文数: 0 引用数: 0
h-index: 0
机构: Department of Chemistry, Columbia University, New York
[8]
Environmental catalysis: trends and outlook
[J].
Centi, G
;
Ciambelli, P
;
Perathoner, S
;
Russo, P
.
CATALYSIS TODAY,
2002, 75 (1-4)
:3-15

Centi, G
论文数: 0 引用数: 0
h-index: 0
机构: Dipartimento Chim Ind & Ingn Mat, I-98166 Messina, Italy

Ciambelli, P
论文数: 0 引用数: 0
h-index: 0
机构: Dipartimento Chim Ind & Ingn Mat, I-98166 Messina, Italy

Perathoner, S
论文数: 0 引用数: 0
h-index: 0
机构: Dipartimento Chim Ind & Ingn Mat, I-98166 Messina, Italy

Russo, P
论文数: 0 引用数: 0
h-index: 0
机构: Dipartimento Chim Ind & Ingn Mat, I-98166 Messina, Italy
[9]
Organic Synthesis "On Water"
[J].
Chanda, Arani
;
Fokin, Valery V.
.
CHEMICAL REVIEWS,
2009, 109 (02)
:725-748

Chanda, Arani
论文数: 0 引用数: 0
h-index: 0
机构:
Scripps Res Inst, Dept Chem, La Jolla, CA 92037 USA Scripps Res Inst, Dept Chem, La Jolla, CA 92037 USA

Fokin, Valery V.
论文数: 0 引用数: 0
h-index: 0
机构:
Scripps Res Inst, Dept Chem, La Jolla, CA 92037 USA Scripps Res Inst, Dept Chem, La Jolla, CA 92037 USA
[10]
Synthesis and biological activities of new checkpoint kinase 1 inhibitors structurally related to granulatimide
[J].
Conchon, Elisabeth
;
Anizon, Fabrice
;
Aboab, Bettina
;
Prudhomme, Michelle
.
JOURNAL OF MEDICINAL CHEMISTRY,
2007, 50 (19)
:4669-4680

Conchon, Elisabeth
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Blaise Pascal, Lab SEESIB, CNRS, UMR 6504, F-63177 Aubiere, France Univ Blaise Pascal, Lab SEESIB, CNRS, UMR 6504, F-63177 Aubiere, France

Anizon, Fabrice
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Blaise Pascal, Lab SEESIB, CNRS, UMR 6504, F-63177 Aubiere, France Univ Blaise Pascal, Lab SEESIB, CNRS, UMR 6504, F-63177 Aubiere, France

Aboab, Bettina
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Blaise Pascal, Lab SEESIB, CNRS, UMR 6504, F-63177 Aubiere, France Univ Blaise Pascal, Lab SEESIB, CNRS, UMR 6504, F-63177 Aubiere, France

Prudhomme, Michelle
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Blaise Pascal, Lab SEESIB, CNRS, UMR 6504, F-63177 Aubiere, France Univ Blaise Pascal, Lab SEESIB, CNRS, UMR 6504, F-63177 Aubiere, France