Efficient synthesis of substituted imidazo[4,5-b] pyridines

被引：0

作者：

Xing, Yuan-Yuan ^{[1
]}

Liu, Chuanxiang ^{[1
]}

Wu, Fanhong ^{[1
]}

机构：

[1] Shanghai Inst Technol, Sch Chem & Environm Engn, Shanghai 201418, Peoples R China

来源：

HETEROCYCLIC COMMUNICATIONS | 2013年 / 19卷 / 05期

关键词：

cyclization; imidazo[4,5-b]pyridine; synthesis; AGENTS;

D O I：

10.1515/hc-2013-0059

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient approach to the synthesis of 1-methylimidazo[4,5-b]pyridine derivatives 5-10 of biological interest has been developed. The key intermediate product 4 is obtained by cyclization of 2-amino-3-methyl-aminopyridine (3) with phenylacetic acid.

引用

页码：327 / 330

页数：4

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