Efficient synthesis of substituted imidazo[4,5-b] pyridines

被引：0
|
作者：
Xing, Yuan-Yuan [1 ]
Liu, Chuanxiang [1 ]
Wu, Fanhong [1 ]
机构：
[1] Shanghai Inst Technol, Sch Chem & Environm Engn, Shanghai 201418, Peoples R China
来源：
HETEROCYCLIC COMMUNICATIONS | 2013年 / 19卷 / 05期
关键词：
cyclization; imidazo[4,5-b]pyridine; synthesis; AGENTS;
D O I：
10.1515/hc-2013-0059
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
An efficient approach to the synthesis of 1-methylimidazo[4,5-b]pyridine derivatives 5-10 of biological interest has been developed. The key intermediate product 4 is obtained by cyclization of 2-amino-3-methyl-aminopyridine (3) with phenylacetic acid.
引用
收藏
页码：327 / 330
页数：4
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