Solvent-free one-pot synthesis of highly functionalized benzothiazolediamides via Ugi four-component reaction

被引：0

作者：

Sheikholeslami-Farahani, F. ^{[1
]}

Shahvelayati, A. S. ^{[2
]}

机构：

[1] Islamic Azad Univ, Firoozkooh Branch, Dept Chem, Firoozkooh, Iran

[2] Islamic Azad Univ, Dept Chem, Shahre E Rey Branch, Tehran, Iran

来源：

BULGARIAN CHEMICAL COMMUNICATIONS | 2015年 / 47卷 / 03期

关键词：

Ugi reaction; One-pot; Maleic anhydride; 2-Aminobenzothiazole; Solvent-free; MULTICOMPONENT REACTIONS; ALPHA-AMINO; ISOCYANIDE; DISCOVERY; PEPTIDES;

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

4-Benzothiazol-2-ylamino-4-oxo-2-butenoic acid, prepared by reaction of 2-aminobenzothiazole and maleic anhydride, is used as an acid component in Ugi reaction, under solvent-free conditions, to produce unsaturated alpha-benzothiazoleamidodipeptides in good yields using a tandem sequence.

引用

页码：830 / 836

页数：7

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