Facile construction of functionalized 4H-chromene via tandem benzylation and cyclization

被引：80
作者：
Fan, Jinmin
Wang, Zhiyong [1 ]
机构：
[1] Univ Sci & Technol China, Joint Lab Green Synthet Chem, Hefei Natl Lab Phys Sci Microscale, Hefei 230026, Peoples R China
来源：
CHEMICAL COMMUNICATIONS | 2008年 / 42期
基金：
中国国家自然科学基金;
关键词：
D O I：
10.1039/b812046c
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
A series of functionalized 4H-chromenes have been constructed by using a novel FeCl3-catalyzed benzylation-cyclization tandem reaction.
引用
收藏
页码：5381 / 5383
页数：3
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共 29 条
  • [1] Domino reactions of 1,3-bis-silyl enol ethers with benzopyrylium triflates:: Efficient synthesis of fluorescent 6H-benzo[c]chromen-6-ones, dibenzo[c,d]chromen-6-ones, and 2,3-dihydro-1H-4,6-dioxachrysen-5-ones
    Appel, B
    Saleh, NNR
    Langer, P
    [J]. CHEMISTRY-A EUROPEAN JOURNAL, 2006, 12 (04) : 1221 - 1236
  • [2] ANTIINFLAMMATORY MECHANISM OF CORDIACHROMENE-A ACTION
    BENSLIMANE, AF
    POUCHUS, YF
    VERBIST, JF
    PETIT, JY
    BRION, JD
    WELIN, L
    [J]. JOURNAL OF CLINICAL PHARMACOLOGY, 1995, 35 (03) : 298 - 301
  • [3] ENANTIOSELECTIVE TOTAL SYNTHESIS OF MIROESTROL
    COREY, EJ
    WU, LI
    [J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1993, 115 (20) : 9327 - 9328
  • [4] Rhodomyrtone, an antibiotic from Rhodomyrtus tomentosa
    Dachriyanus
    Salni
    Sargent, MV
    Skelton, BW
    Soediro, I
    Sutisna, M
    White, AH
    Yulinah, E
    [J]. AUSTRALIAN JOURNAL OF CHEMISTRY, 2002, 55 (03) : 229 - 232
  • [5] O-arylation versus C-arylation: Copper-catalyzed intramolecular coupling of aryl bromides with 1,3-dicarbonyls
    Fang, Yewen
    Li, Chaozhong
    [J]. JOURNAL OF ORGANIC CHEMISTRY, 2006, 71 (17) : 6427 - 6431
  • [6] Reactions of salicyl N-tosylimines or salicylaldehydes with diethyl acetylenedicarboxylate for the synthesis of highly functionalized chromenes
    Guo, Ying-Wen
    Shi, Yong-Ling
    Li, Hong-Bin
    Shi, Min
    [J]. TETRAHEDRON, 2006, 62 (25) : 5875 - 5882
  • [7] Discovery of potent chromen-4-one inhibitors of the DNA-dependent protein kinase (DNA-PK) using a small-molecule library approach
    Hardcastle, IR
    Cockcroft, X
    Curtin, NJ
    El-Murr, MD
    Leahy, JJJ
    Stockley, M
    Golding, BT
    Rigoreau, L
    Richardson, C
    Smith, GCM
    Griffin, RJ
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 2005, 48 (24) : 7829 - 7846
  • [8] An efficient and general iron-catalyzed arylation of benzyl alcohols and benzyl carboxylates
    Iovel, I
    Mertins, K
    Kischel, J
    Zapf, A
    Beller, M
    [J]. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2005, 44 (25) : 3913 - 3917
  • [9] Aqua mediated synthesis of substituted 2-amino-4H-chromenes and in vitro study as antibacterial agents
    Kidwai, M
    Saxena, S
    Khan, MKR
    Thukral, SS
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2005, 15 (19) : 4295 - 4298
  • [10] A general and efficient iron-catalyzed benzylation of 1,3-dicarbonyl compounds
    Kischel, Jette
    Mertins, Kristin
    Michalik, Dirk
    Zapf, Alexander
    Beller, Matthias
    [J]. ADVANCED SYNTHESIS & CATALYSIS, 2007, 349 (06) : 865 - 870
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