Synthesis and evaluation of a new PET ligand for imaging of monoacylglycerol lipase in brain

被引：0
|
作者：
Mori, Wakana [1 ]
Kurihara, Yusuke [2 ]
Hatori, Akiko [1 ]
Zhang, Yiding [1 ]
Fujinaga, Masayuki [1 ]
Zhang, Ming-Rong [1 ]
机构：
[1] Natl Inst Quantum & Radiol Sci & Technol, Dept Radiopharmaceut Dev, Natl Inst Radiol Sci, Chiba, Japan
[2] SHI Accelerator Serv, Tokyo, Japan
来源：
JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 2019年 / 62卷
关键词：
PRECLINICAL EVALUATION;
D O I：
暂无
中图分类号：
Q5 [生物化学];
学科分类号：
071010 ; 081704 ;
摘要：
P-238
引用
收藏
页码：S394 / S395
页数：2
相关论文
共 50 条
  • [21] Rapid synthesis and in vitro and in vivo evaluation of folic acid derivatives labeled with fluorine-18 for PET imaging of folate receptor-positive tumors
    Al Jammaz, I.
    Al-Otaibi, B.
    Amer, S.
    Okarvi, S. M.
    NUCLEAR MEDICINE AND BIOLOGY, 2011, 38 (07) : 1019 - 1028
  • [22] Synthesis, Structure-Activity Relationships, Radiofluorination, and Biological Evaluation of [18F]RM365, a Novel Radioligand for Imaging the Human Cannabinoid Receptor Type 2 (CB2R) in the Brain with PET
    Teodoro, Rodrigo
    Gundel, Daniel
    Deuther-Conrad, Winnie
    Kazimir, Aleksandr
    Toussaint, Magali
    Wenzel, Barbara
    Bormans, Guy
    Hey-Hawkins, Evamarie
    Kopka, Klaus
    Brust, Peter
    Moldovan, Rares Petru
    JOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (20) : 13991 - 14010
  • [23] Radiolabeled new somatostatin analogs conjugated to DOMA chelator used as targeted tumor imaging agent: synthesis and radiobiological evaluation
    De, Kakali
    Banerjee, Indranil
    Misra, Mridula
    AMINO ACIDS, 2015, 47 (06) : 1135 - 1153
  • [24] Synthesis and Preliminary Evaluation of a New 99mTc Labeled Substance P Analogue as a Potential Tumor Imaging Agent
    Mozaffari, Saeed
    Erfani, Mostafa
    Beiki, Davood
    Daha, Fariba Johari
    Kobarfard, Farzad
    Balalaie, Saeed
    Fallahi, Babak
    IRANIAN JOURNAL OF PHARMACEUTICAL RESEARCH, 2015, 14 (01): : 97 - 110
  • [25] (R)-[18F]NEBIFQUINIDE: A promising new PET tracer for TSPO imaging
    Berroteran-Infante, Neydher
    Kalina, Thomas
    Fetty, Lukas
    Janisch, Victoria
    Velasco, Ramona
    Vraka, Chrysoula
    Hacker, Marcus
    Haug, Alexander R.
    Pallitsch, Katharina
    Wadsak, Wolfgang
    Mitterhauser, Markus
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 176 : 410 - 418
  • [26] Design, Synthesis, and Biological Evaluation of Polyaminocarboxylate Ligand-Based Theranostic Conjugates for Antibody-Targeted Cancer Therapy and Near-Infrared Optical Imaging
    Ren, Siyuan
    Sun, Xiang
    Wang, Haixing
    Trung Hai Nguyen
    Sadeghipour, Negar
    Xu, Xiaochun
    Kang, Chi Soo
    Liu, Yujie
    Xu, Hua
    Wu, Ningjie
    Chen, Yanda
    Tichauer, Kenneth
    Minh, David D. L.
    Chong, Hyun-Soon
    CHEMMEDCHEM, 2018, 13 (24) : 2606 - 2617
  • [27] Development of [18F]LU14 for PET Imaging of Cannabinoid Receptor Type 2 in the Brain
    Teodoro, Rodrigo
    Guendel, Daniel
    Deuther-Conrad, Winnie
    Ueberham, Lea
    Toussaint, Magali
    Bormans, Guy
    Brust, Peter
    Moldovan, Rares-Petru
    INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2021, 22 (15)
  • [28] Novel Thienopyrimidine-Based PET Tracers for P2Y12 Receptor Imaging in the Brain
    van der Wildt, Berend
    Janssen, Bieneke
    Pekosak, Aleksandra
    Steen, E. Johanna L.
    Schuit, Robert C.
    Kooijman, Esther J. M.
    Beaino, Wissam
    Vugts, Danielle J.
    Windhorst, Albert D.
    ACS CHEMICAL NEUROSCIENCE, 2021, 12 (23): : 4465 - 4474
  • [29] Development of a New Folate-Derived Ga-68-Based PET Imaging Agent
    Brand, Christian
    Longo, Valerie A.
    Groaning, Mike
    Weber, Wolfgang A.
    Reiner, Thomas
    MOLECULAR IMAGING AND BIOLOGY, 2017, 19 (05) : 754 - 761
  • [30] Synthesis and evaluation of a ligand targeting the somatostatin-2 receptor for drug delivery to neuroendocrine cancers
    Li, Guo
    Low, Philip S.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 25 (08) : 1792 - 1798
12345