Highly diastereoselective synthesis of N-protected arylglycine derivatives via TiCl4-promoted Friedel-Crafts reaction of phenols with chiral N,O-hemiacetal

被引:0
作者
Ge, CS [1 ]
Chen, YJ [1 ]
Wang, D [1 ]
机构
[1] Chinese Acad Sci, Inst Chem, Ctr Mol Sci, Beijing 100080, Peoples R China
关键词
Friedel-Crafts reaction; arylglycine; chiral N; O-hemiacetal;
D O I
暂无
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
The optically active N-protected arylglycine derivatives were obtained via TiCl4-promoted Friedel-Crafts reaction of various phenols with chiral N,O-hemiacetals in excellent diastereoselectivity.
引用
收藏
页码:37 / 42
页数:6
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