Synthesis and fungicidal activity of new fluorine-containing mandelic acid amide compounds

被引：16

作者：

Li, Shuai ^{[1
]}

Cui, Can ^{[1
]}

Wang, Man-Yi ^{[1
]}

Yu, Shui-Jing ^{[1
]}

Shi, Yan-Xia ^{[2
]}

Zhang, Xiao ^{[1
]}

Li, Zheng-Ming ^{[1
]}

Zhao, Wei-Guang ^{[1
]}

Li, Bao-Ju ^{[2
]}

机构：

[1] Nankai Univ, Natl Pesticide Engn Res Ctr Tianjin, State Key Lab Elementoorgan Chem, Tianjin 300071, Peoples R China

[2] Chinese Acad Agr Sci, Inst Vegetables & Flowers, Beijing 100193, Peoples R China

来源：

JOURNAL OF FLUORINE CHEMISTRY | 2012年 / 137卷

基金：

中国国家自然科学基金;

关键词：

Fluorinated mandelic acid amide; Fungicidal activities; Synthesis; DRUGS;

D O I：

10.1016/j.jfluchem.2012.02.011

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

A series of novel fluorine-containing mandelic acid amide compounds were designed and synthesized by a facile method, and their structures were characterized by H-1 nuclear magnetic resonance (NMR) and high-resolution mass spectrometry. The preliminary in vivo bioassays indicated that some of the title compounds showed excellent fungicidal activities in vivo against Pseudoperonospora cubensis at the dosage of 25 mg L-1, which were comparable with the control (Mandipropamid). (c) 2012 Elsevier B.V. All rights reserved.

引用

页码：108 / 112

页数：5

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