Application of polymer-bound phosphonium salts as traceless supports for solid phase synthesis

被引：101

作者：

Hughes, I

机构：

[1] SmithKline Beecham Pharmaceuticals, New Frontiers Science Park (North), Harlow CM19 5AW, Third Avenue

来源：

TETRAHEDRON LETTERS | 1996年 / 37卷 / 42期

关键词：

D O I：

10.1016/0040-4039(96)01669-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The utility of the phosphonium group as a traceless linker for the solid phase synthesis of small organic molecules is demonstrated by the elaboration of polymer-bound phosphonium salts and their subsequent cleavage to alkyl, alkenyl and heteroaryl products. Copyright (C) 1996 Elsevier Science Ltd

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收藏

页码：7595 / 7598

页数：4

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