A rapid and high-yielding synthesis of thiazoles and aminothiazoles using ammonium-12-molybdophosphate

被引：77
作者：
Das, Biswanath [1 ]
Reddy, V. Saidi [1 ]
Ramu, R. [1 ]
机构：
[1] Indian Inst Chem Technol, Organ Chem Div 1, Hyderabad 500007, Andhra Pradesh, India
来源：
JOURNAL OF MOLECULAR CATALYSIS A-CHEMICAL | 2006年 / 252卷 / 1-2期
关键词：
thiazole; aminothiazole; phenacyl bromide; thioamide; thiourea; ammonium-12-molybdophosphate;
D O I：
10.1016/j.molcata.2006.02.065
中图分类号：
O64 [物理化学（理论化学）、化学物理学];
学科分类号：
070304 ; 081704 ;
摘要：
A convenient method for the synthesis of thiazoles and aminothiazoles by treatment of phenacyl bromides with thioamides/thiourea in the presence of ammonium-12-molybdophosphate at room temperature has been developed. The products are formed rapidly (within 20 min) and in excellent yields. (c) 2006 Elsevier B.V. All rights reserved.
引用
收藏
页码：235 / 237
页数：3
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