Synthesis and Antimicrobial Activity of Azolyl Pyrimidines

被引：10

作者：

Butta, Ragavendra ^{[1
]}

Donthamsetty, Sowmya, V ^{[1
]}

Adivireddy, Padmaja ^{[1
]}

Venkatapuram, Padmavathi ^{[1
]}

机构：

[1] Sri Venkateswara Univ, Dept Chem, Tirupati 517502, Andhra Pradesh, India

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2017年 / 54卷 / 01期

关键词：

MARINE SPONGE; DERIVATIVES; ANALOGS; ANTIBACTERIAL; DESIGN; AGENTS; WATER;

D O I：

10.1002/jhet.2615

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A new class of azolyl pyrimidines linked by diamino sulfone moiety was prepared and studied their antimicrobial activity. Chloro-substituted and nitro-substituted thiazolyl pyrimidines (9c and 9e) showed excellent antibacterial activity against Bacillus subtilis, while imidazolyl pyrimidines (10c and 10e) exhibited promising antifungal activity against Aspergillus niger.

引用

页码：524 / 530

页数：7

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