Synthesis and Antimicrobial Activity of Azolyl Pyrimidines

被引：10
作者：
Butta, Ragavendra [1 ]
Donthamsetty, Sowmya, V [1 ]
Adivireddy, Padmaja [1 ]
Venkatapuram, Padmavathi [1 ]
机构：
[1] Sri Venkateswara Univ, Dept Chem, Tirupati 517502, Andhra Pradesh, India
来源：
JOURNAL OF HETEROCYCLIC CHEMISTRY | 2017年 / 54卷 / 01期
关键词：
MARINE SPONGE; DERIVATIVES; ANALOGS; ANTIBACTERIAL; DESIGN; AGENTS; WATER;
D O I：
10.1002/jhet.2615
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A new class of azolyl pyrimidines linked by diamino sulfone moiety was prepared and studied their antimicrobial activity. Chloro-substituted and nitro-substituted thiazolyl pyrimidines (9c and 9e) showed excellent antibacterial activity against Bacillus subtilis, while imidazolyl pyrimidines (10c and 10e) exhibited promising antifungal activity against Aspergillus niger.
引用
收藏
页码：524 / 530
页数：7
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