Development of potent SHP2 inhibitors for in vivo studies

被引:0
|
作者
Ge, Yiyu [1 ]
Lawrence, Harshani R. [1 ]
Chen, Liwei [1 ]
Scott, Latanya M. [1 ]
Sebti, Said M. [1 ]
Lawrence, Nicholas J. [1 ]
Wu, Jie [1 ]
机构
[1] Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL 33612 USA
关键词
D O I
10.1158/1538-7445.AM2012-2912
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
2912
引用
收藏
页数:1
相关论文
共 50 条
  • [31] SHP2 is involved in the occurrence, development and prognosis of cancer
    Li, Shu
    Qu, Jialing
    Wang, Xiaotong
    Zou, Qin
    Li, Chunli
    ONCOLOGY LETTERS, 2023, 26 (03)
  • [32] Shp2 in myocytes is essential for cardiovascular and neointima development
    Gong, Hui
    Ni, Jiaojiao
    Xu, Zhiyong
    Huang, Jiaqi
    Zhang, Jie
    Huang, Yizhou
    Zeng, Chunlai
    Zhang, Xue
    Cheng, Hongqiang
    Ke, Yuehai
    JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY, 2019, 137 : 71 - 81
  • [33] Tyrosine phosphatase SHP2 inhibitors in tumor-targeted therapies
    Zhendong Song
    Meijing Wang
    Yang Ge
    Xue-Ping Chen
    Ziyang Xu
    Yang Sun
    Xiao-Feng Xiong
    Acta Pharmaceutica Sinica B, 2021, 11 (01) : 13 - 29
  • [34] Tyrosine phosphatase SHP2 inhibitors in tumor-targeted therapies
    Song, Zhendong
    Wang, Meijing
    Ge, Yang
    Chen, Xue-Ping
    Xu, Ziyang
    Sun, Yang
    Xiong, Xiao-Feng
    ACTA PHARMACEUTICA SINICA B, 2021, 11 (01) : 13 - 29
  • [35] Recent advances in the discovery of protein tyrosine phosphatase SHP2 inhibitors
    Kong, Jiao
    Long, Ya-Qiu
    RSC MEDICINAL CHEMISTRY, 2022, 13 (03): : 246 - 257
  • [36] A patent review of SHP2 allosteric inhibitors (2018-present)
    Petrocchi, Alessia
    Ciammaichella, Alina
    EXPERT OPINION ON THERAPEUTIC PATENTS, 2024, 34 (05) : 383 - 396
  • [37] MEDI 305-Inhibitors of SHP2, a protein tyrosine phosphatase
    Ramamoorthy, Divya
    Pireddu, Roberta
    He, Jing
    Wu, Xin
    Luo, Yunting
    Lawrence, Harshani R.
    Sung, Shen-Shu
    Chen, LiWei
    Sebti, Said M.
    Wu, Jerry
    Lawrence, Nicholas J.
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2008, 236
  • [38] Discovery of a SHP2 Degrader with In Vivo Anti-Tumor Activity
    Miao, Jinmin
    Bai, Yunpeng
    Miao, Yiming
    Qu, Zihan
    Dong, Jiajun
    Zhang, Ruo-Yu
    Aggarwal, Devesh
    Jassim, Brenson A.
    Nguyen, Quyen
    Zhang, Zhong-Yin
    MOLECULES, 2023, 28 (19):
  • [39] Functions of Shp2 in cancer
    Zhang, Jie
    Zhang, Fei
    Niu, Ruifang
    JOURNAL OF CELLULAR AND MOLECULAR MEDICINE, 2015, 19 (09) : 2075 - 2083
  • [40] Phosphorylation of SHP2 at Tyr62 Enables Acquired Resistance to SHP2 Allosteric Inhibitors in FLT3-ITD-Driven AML
    Pfeiffer, Anamarija
    Franciosa, Giulia
    Locard-Paulet, Marie
    Piga, Ilaria
    Reckzeh, Kristian
    Vemulapalli, Vidyasiri
    Blacklow, Stephen C.
    Theilgaard-Monch, Kim
    Jensen, Lars J.
    V. Olsen, Jesper
    CANCER RESEARCH, 2022, 82 (11) : 2141 - 2155