Synthesis of maleopimaric and citraconopimaric acids N-[3-(pyrimidin-2-yl)aryl]amides

被引：2
|
作者：
Koroleva, E. V. [1 ]
Gusak, K. N. [1 ]
Ignatovich, Zh V. [1 ]
Ermolinskaya, A. L. [1 ]
Bei, M. P. [1 ]
Yuvchenko, A. P. [1 ]
机构：
[1] Acad Sci Belarus, Inst New Mat Chem, Natl Acad Belarus, Minsk 220141, BELARUS
来源：
RUSSIAN JOURNAL OF ORGANIC CHEMISTRY | 2012年 / 48卷 / 08期
关键词：
DERIVATIVES;
D O I：
10.1134/S1070428012080143
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Acylation of 6-methyl-N-[4-(pyridin-3-yl)pyrimidin-2-yl]benzene-1,3-diamine, 4-methyl-N-[4-(pyridin-3-yl)pyrimidin-2-yl]benzene-1,3-diamine, and N-[4-(pyridin-3-yl)pyrimidin-2-yl]benzene-1,3-diamine with maleopimaric and citraconopimaric acid chlorides, with benzotriazolyl maleopimarate afforded N-[3-(pyrimidin-2-yl)aryl]amides of maleopimaric and citraconopimaric acids. By the reaction of substituted N-arylamides of maleopimaric acid with methanesulfonic acid biologically active methanesulfonates were obtained.
引用
收藏
页码：1121 / 1125
页数：5
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