Synthesis of maleopimaric and citraconopimaric acids N-[3-(pyrimidin-2-yl)aryl]amides

被引：2

作者：

Koroleva, E. V. ^{[1
]}

Gusak, K. N. ^{[1
]}

Ignatovich, Zh V. ^{[1
]}

Ermolinskaya, A. L. ^{[1
]}

Bei, M. P. ^{[1
]}

Yuvchenko, A. P. ^{[1
]}

机构：

[1] Acad Sci Belarus, Inst New Mat Chem, Natl Acad Belarus, Minsk 220141, BELARUS

来源：

RUSSIAN JOURNAL OF ORGANIC CHEMISTRY | 2012年 / 48卷 / 08期

关键词：

DERIVATIVES;

D O I：

10.1134/S1070428012080143

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Acylation of 6-methyl-N-[4-(pyridin-3-yl)pyrimidin-2-yl]benzene-1,3-diamine, 4-methyl-N-[4-(pyridin-3-yl)pyrimidin-2-yl]benzene-1,3-diamine, and N-[4-(pyridin-3-yl)pyrimidin-2-yl]benzene-1,3-diamine with maleopimaric and citraconopimaric acid chlorides, with benzotriazolyl maleopimarate afforded N-[3-(pyrimidin-2-yl)aryl]amides of maleopimaric and citraconopimaric acids. By the reaction of substituted N-arylamides of maleopimaric acid with methanesulfonic acid biologically active methanesulfonates were obtained.

引用

页码：1121 / 1125

页数：5