Structure based design and synthesis of novel orally active thrombin inhibitors

被引:0
作者
Haramura, M [1 ]
Shiraishi, T [1 ]
Haneishi, T [1 ]
Kuromaru, K [1 ]
Ohta, M [1 ]
Kim, JM [1 ]
Nam, WH [1 ]
Jung, KY [1 ]
Jeon, GH [1 ]
Kozono, T [1 ]
机构
[1] Chugai Pharmaceut Co Ltd, Chem Res Lab, Shizuoka 412, Japan
来源
PEPTIDE SCIENCE - PRESENT AND FUTURE | 1999年
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:639 / 641
页数:3
相关论文
共 4 条
[1]  
BURTON PS, 1991, ADV DRUG DELIVER REV, V7, P365, DOI 10.1016/0169-409X(91)90014-4
[2]   ARGATROBAN, A SELECTIVE, POTENT THROMBIN INHIBITOR [J].
BUSH, LR .
CARDIOVASCULAR DRUG REVIEWS, 1991, 9 (03) :247-263
[3]  
GOULD RJ, 1993, PERSPECT DRUG DISCOV, V1, P419
[4]  
STUBBS MT, 1993, PERSPECT DRUG DISCOV, V1, P431