Construction of a Library of Arylpiperazinyl 1,2,3-Triazole Derivatives as Ligands for Dopamine D3/D4 Receptor

被引：3

作者：

Kwak, Ju Myung ^{[1
]}

Moon, Ji Soo ^{[1
]}

Choi, Jea I. ^{[1
]}

Murugan, Ravichandran N. ^{[4
]}

Park, Woo Kyu ^{[2
]}

Gong, Jae Yang ^{[3
]}

Lee, Hee Yoon ^{[4
]}

Koh, Hun Yeong ^{[1
]}

机构：

[1] Inha Univ, Dept Chem, Inchon 402751, South Korea

[2] Korea Res Inst Chem Technol, Pharmaceut Screening Res Team, Taejon 305343, South Korea

[3] Keimyung Univ, Coll Pharm, Taegu 704701, South Korea

[4] Korea Adv Inst Sci & Technol, Dept Chem, Taejon 305701, South Korea

来源：

BULLETIN OF THE KOREAN CHEMICAL SOCIETY | 2013年 / 34卷 / 11期

关键词：

Dopamine receptor ligand; 1,2,3-Triazole; Arylpiperazine; Heterocyclization; Microwave reaction; POTENT; CYCLOADDITION; LEAD;

D O I：

10.5012/bkcs.2013.34.11.3467

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

[No abstract available]

引用

页码：3467 / 3470

页数：4

共 33 条

[1] DIPOLAR CYCLO-ADDITION REACTIONS OF ORGANIC AZIDES WITH SOME ACETYLENIC-COMPOUNDS [J].

ABUORABI, ST ;

ATFAH, MA ;

JIBRIL, I ;

MARII, FM ;

ALI, AAS .

JOURNAL OF HETEROCYCLIC CHEMISTRY, 1989, 26 (05) :1461-1468

[2] Recent developments in microwave-assisted, transition-metal-catalysed C-C and C-N bond-forming reactions [J].

Appukkuttan, Prasad ;

Van der Eycken, Erik .

EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2008, 2008 (07) :1133-1155

[3]

BRESLOW R, 1998, WATER SOLVENT CHEM R

[4] Design of novel hexahydropyrazinoquinolines as potent and selective dopamine D3 receptor ligands with improved solubility [J].

Chen, JY ;

Ding, K ;

Levant, B ;

Wang, SM .

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2006, 16 (02) :443-446

[5] The use of bioisosteric groups in lead optimization [J].

Chen, XQ ;

Wang, WB .

ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 38, 2003, 38 :333-346

[6] Microwave energy: a versatile tool for the biosciences [J].

Collins, Jonathan M. ;

Leadbeater, Nicholas E. .

ORGANIC & BIOMOLECULAR CHEMISTRY, 2007, 5 (08) :1141-1150

[7] Microwave-assisted synthesis in water as solvent [J].

Dallinger, Doris ;

Kappe, C. Oliver .

CHEMICAL REVIEWS, 2007, 107 (06) :2563-2591

[8] 2-[(4-phenylpiperazin-1-yl)methyl]imidazo(di)azines as selective D4-ligands.: Induction of penile erection by 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a potent and selective D4 partial agonist [J].

Enguehard-Gueiffier, Cecile ;

Huebner, Harald ;

El Hakmaoui, Ahmed ;

Allouchi, Hassan ;

Gmeiner, Peter ;

Argiolas, Antonio ;

Melis, Maria Rosaria ;

Gueiffier, Alain .

JOURNAL OF MEDICINAL CHEMISTRY, 2006, 49 (13) :3938-3947

[9]

Grieco P.A., 1998, Organic Synthesis in Water

[10] Reactions of C-H bonds in water [J].

Herrerias, Clara I. ;

Yao, Xiaoquan ;

Li, Zhiping ;

Li, Chao-Jun .

CHEMICAL REVIEWS, 2007, 107 (06) :2546-2562

← 1 2 3 4 →