Facile entry to 4-and 5-hydroxybenzofuran and to their amino derivatives

被引:21
作者
Bonini, Carlo [1 ]
Cristiani, Graziella [1 ]
Funicello, Maria [1 ]
Viggiani, Licia [1 ]
机构
[1] Univ Basilicata, Dept Chem, I-85100 Potenza, Italy
关键词
aminobenzo condensed derivatives; 4-hydroxybenzofuran; smiles rearrangement;
D O I
10.1080/00397910600634118
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
An innovative one-step procedure for the synthesis of 4-hydroxybenzofuran and an improved synthesis of 5-hydroxybenzofuran is reported. Such compounds were also transformed into their amino derivatives via Smiles rearrangement with good to high overall yields.
引用
收藏
页码:1983 / 1990
页数:8
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