Synthesis and Herbicidal Activity of Amide Derivatives Containing Thiazole Moiety

被引：7

作者：

Weng, Jian-Quan ^{[1
]}

Liu, Xing-Hai ^{[1
]}

Tong, Guo-Tong ^{[2
]}

机构：

[1] Zhejiang Univ Technol, Coll Chem Engn & Mat Sci, Hangzhou 310014, Zhejiang, Peoples R China

[2] Hangzhou Vocat & Tech Coll, Dept Chem Engn, Hangzhou 310018, Zhejiang, Peoples R China

来源：

ASIAN JOURNAL OF CHEMISTRY | 2013年 / 25卷 / 04期

基金：

中国国家自然科学基金;

关键词：

Synthesis; Amide derivative; Thiazole; Herbicidal activity; BIOLOGICAL-ACTIVITIES; ANALOGS;

D O I：

10.14233/ajchem.2013.13366

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Twelve novel amide derivatives containing thiazole moiety were synthesized via a coupling reaction of [4-(substituted phenypthiazol-2-yl] acetonitrile and aryl isocyanates catalyzed by organic bases. Their structures were characterized by H-1 NMR, FTIR, MS and elemental analysis. The preliminary bioassay indicated that these compounds exhibited moderate herbicidal activities against Echinochloa crusgalli and Amaranthus ascedense.

引用

页码：2149 / 2152

页数：4

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