Synthesis and characterization of novel 1,2,3-triazole-linked theophylline and coumarin s-triazines

被引:0
作者
Joshi, Penny [1 ,2 ]
Tripathi, Mohit [1 ]
Rawat, Diwan S. [1 ]
机构
[1] Univ Delhi, Dept Chem, Delhi 110007, India
[2] Kumaun Univ, Dept Chem, Naini Tal 263001, India
来源
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 2014年 / 53卷 / 03期
关键词
s-Triazine; dendrimer; triazole; theophylline; coumarin; VITRO ANTIMALARIAL ACTIVITY; IMPROVED IN-VITRO; ANTIBACTERIAL ACTIVITY; DRUG-DELIVERY; DERIVATIVES; HYBRIDS; CYTOTOXICITY; DENDRIMERS; ANALOGS; DESIGN;
D O I
暂无
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
A series of novel s-triazine-1,2,3-triazole-theophylline and s-triazine-1,2,3-triazole-coumarin generation-0 dendrimers has been synthesized and characterized by FT-IR, H-1 and C-13 NMR, and mass-spectral methods. Some 'selected compounds have been evaluated for antibacterial and antifungal activity against a variety of strains and for anti-cancer activity against 60 human cancer cell lines.
引用
收藏
页码:311 / 318
页数:8
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