Highly diastereoselective radical cyclisations of chiral sulfinimines

被引:23
作者
Rochette, Elise M. [1 ]
Lewis, William [1 ]
Dossetter, Al G. [2 ]
Stockman, Robert A. [1 ]
机构
[1] Univ Nottingham, Sch Chem, Nottingham NG7 2RD, England
[2] AstraZeneca, Macclesfield SK10 4TG, Cheshire, England
基金
英国工程与自然科学研究理事会;
关键词
ASYMMETRIC-SYNTHESIS; ALDIMINES; EFFICIENT; ALCOHOLS; IMINES;
D O I
10.1039/c3cc45452e
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
Chiral amines are formed by the highly diastereoselective intramolecular addition of alkyl and aryl radicals onto chiral mesityl sulfinimines.
引用
收藏
页码:9395 / 9397
页数:3
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