共 50 条
- [1] MEDI 54-Syntheses and SAR of piperidin-3-yl ureas as potent and selective 11β-HSD-1 inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2007, 234Li, Yun-Long论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Expt Stn E336, Wilmington, DE 19880 USA Incyte Corp, Expt Stn E336, Wilmington, DE 19880 USABostrom, Lori论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Expt Stn E336, Wilmington, DE 19880 USA Incyte Corp, Expt Stn E336, Wilmington, DE 19880 USAZhuo, Jincong论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Expt Stn E336, Wilmington, DE 19880 USA Incyte Corp, Expt Stn E336, Wilmington, DE 19880 USALi, Yanlong论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Expt Stn E336, Wilmington, DE 19880 USA Incyte Corp, Expt Stn E336, Wilmington, DE 19880 USACovington, Maryanne论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Incyte Corp, Expt Stn E336, Wilmington, DE 19880 USAHuber, Reid论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Expt Stn E336, Wilmington, DE 19880 USA Incyte Corp, Expt Stn E336, Wilmington, DE 19880 USAMetcalf, Brian论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Expt Stn E336, Wilmington, DE 19880 USA Incyte Corp, Expt Stn E336, Wilmington, DE 19880 USAYao, Wenqing论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Expt Stn E336, Wilmington, DE 19880 USA Incyte Corp, Expt Stn E336, Wilmington, DE 19880 USA
- [2] MEDI 402-Discovery of potent and selective 11ß-HSD-1 inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2006, 232Patel, Jyoti R.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, GPRD, Abbott Pk, IL 60064 USAShuai, Qi论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, GPRD, Abbott Pk, IL 60064 USADinges, Jurgen论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, GPRD, Abbott Pk, IL 60064 USAWinn, Martin论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, GPRD, Abbott Pk, IL 60064 USAPliushchev, Marina论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, GPRD, Abbott Pk, IL 60064 USAFung, Steven论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, GPRD, Abbott Pk, IL 60064 USAMonzon, Katina论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, GPRD, Abbott Pk, IL 60064 USAWang, Jiahong论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, GPRD, Abbott Pk, IL 60064 USAChiou, William J.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, GPRD, Abbott Pk, IL 60064 USAPan, Liping论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, GPRD, Abbott Pk, IL 60064 USALongenecker, Kenton论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, GPRD, Abbott Pk, IL 60064 USAShaml, Hing论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, GPRD, Abbott Pk, IL 60064 USAJacobsonl, Peer论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, GPRD, Abbott Pk, IL 60064 USALink, J. T.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, GPRD, Abbott Pk, IL 60064 USA
- [3] MEDI 48-Discovery and synthesis of nipecotic amide as novel, potent and selective 11ß-HSD-1 inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2007, 234Zhuo, Jincong论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USA Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USAXu, Meizhong论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USA Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USAZhang, Colin论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USA Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USAQian, Dingquan论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USA Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USALi, Yanlong论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USA Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USAHuber, Reid论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USA Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USACovington, Maryanne论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USAMarando, Cindy论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USA Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USAMetcalf, Brian论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USA Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USAYao, Wenqing论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USA Incyte Corp, Expt Stn E336 208B, Wilmington, DE 19880 USA
- [4] Discovery of adamantane ethers as inhibitors of 11β-HSD-1:: Synthesis and biological evaluationBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2007, 17 (03) : 750 - 755Patel, Jyoti R.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAShuai, Qi论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USADinges, Jurgen论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAWinn, Marty论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAPliushchev, Marina论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAFung, Steven论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAMonzon, Katina论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAChiou, William论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAWang, Jiahong论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAPan, Liping论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAWagaw, Seble论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAEngstrom, Kenneth论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAKerdesky, Francis A.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USALongenecker, Kenton论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAJudge, Russell论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAQin, Wenying论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAImade, Hovis M.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAStolarik, DeAnne论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USABeno, David W. A.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USABrune, Michael论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAChovan, Linda E.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USASham, Hing L.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAJacobson, Peer论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USALink, J. T.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA
- [5] Discovery of potent and selective inhibitors of 11β-HSD1 for the treatment of metabolic syndromeBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2006, 16 (24) : 6241 - 6245Richards, Steven论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USASorensen, Bryan论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USAJae, Hwan-Soo论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USAWinn, Marty论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USAChen, Yixian论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USAWang, Jiahong论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USAFung, Steven论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USAMonzon, Katina论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USAFrevert, Ernst U.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USAJacobson, Peer论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USASham, Hing论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USALink, J. T.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, Metabol Dis Res, GPRD, Abbott Pk, IL 60064 USA
- [6] Discovery of N-(piperidin-3-yl)-N-(pyridin-2-yl)piperidine/piperazine-1-carboxamides as small molecule inhibitors of PCSK9BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 28 (23-24) : 3685 - 3688Londregan, Allyn T.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USAAspnes, Gary论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USALimberakis, Chris论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USALoria, Paula M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USAMcClure, Kim F.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USAPetersen, Donna N.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USARaymer, Brian论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USARuggeri, Roger B.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USAWei, Liuqing论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USAXiao, Jun论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USAPiotrowski, David W.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USA Pfizer Inc, Pfizer Med Chem, Eastern Point Rd, Groton, CT 06340 USA
- [7] MEDI 257-Discovery of hydroxyisoquinolines as novel and potent 11-β-HSD-1 inhibitors for the treatment of type 2 diabetesABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2008, 236Wu, Shung C.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAYoon, David S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAVan Kirk, Katy论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Early Discovery Chem, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAPadmanabha, Ramesh论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USACook, Lynda S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USANayeem, Akbar论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Comp Assisted Drug Design, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAGordon, David论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Res, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USASeethala, Ramakrishna论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Res, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAGolla, Rajasree论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Res, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAHosagrahara, Vinayak论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Metab & Pharmacokinet, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAZhang, Lisa论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Metab & Pharmacokinet, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAWang, Meng Meng论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Metab & Pharmacokinet, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USASleczka, Bogdan论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Metab & Pharmacokinet, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAHarper, Timothy论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Metab & Pharmacokinet, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAHarrity, Thomas论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Biol, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USATaylor, Joseph论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Biol, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAPoticello, Randolph论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Biol, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAZebo, Rachel论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Biol, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAMorgan, Nathan论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Biol, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAKirby, Mark S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Res, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USABin, He论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Res, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAKnox, Ronald J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAZvyaga, Tatyana论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Biol, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USAShou, Wilson论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Metab Dis Biol, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USALi, Yi-Xin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Analyt Sci, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USARobl, Jeffery A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Princeton, NJ 08543 USA
- [8] Design, synthesis, and SAR studies of novel polycyclic acids as potent and selective inhibitors of human 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD-1)BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (22) : 6699 - 6704Ye, Xiang-Yang论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Chem, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem, Res & Dev, Princeton, NJ 08543 USAChen, Stephanie Y.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Chem, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem, Res & Dev, Princeton, NJ 08543 USANayeem, Akbar论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, CADD, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem, Res & Dev, Princeton, NJ 08543 USAGolla, Rajasree论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Lead Evaluat, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem, Res & Dev, Princeton, NJ 08543 USASeethala, Ramakrishna论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Lead Evaluat, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem, Res & Dev, Princeton, NJ 08543 USAWang, Mengmeng论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, MAP, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem, Res & Dev, Princeton, NJ 08543 USAHarper, Timothy论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, MAP, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem, Res & Dev, Princeton, NJ 08543 USASleczka, Bogdan G.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, BDAS, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem, Res & Dev, Princeton, NJ 08543 USALi, Yi-Xin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, BDAS, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem, Res & Dev, Princeton, NJ 08543 USAHe, Bin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Biol, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem, Res & Dev, Princeton, NJ 08543 USAKirby, Mark论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Biol, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem, Res & Dev, Princeton, NJ 08543 USAGordon, David A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Biol, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem, Res & Dev, Princeton, NJ 08543 USARobl, Jeffrey A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Chem, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem, Res & Dev, Princeton, NJ 08543 USA
- [9] The discovery of azepane sulfonamides as potent 11β-HSD1 inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 19 (16) : 4563 - 4565Neelamkavil, Santhosh F.论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Corp, Res Inst, Kenilworth, NJ 07033 USA Schering Plough Corp, Res Inst, Kenilworth, NJ 07033 USABoyle, Craig D.论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Corp, Res Inst, Kenilworth, NJ 07033 USA Schering Plough Corp, Res Inst, Kenilworth, NJ 07033 USAChackalamannil, Samuel论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Corp, Res Inst, Kenilworth, NJ 07033 USA Schering Plough Corp, Res Inst, Kenilworth, NJ 07033 USAGreenlee, William J.论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Corp, Res Inst, Kenilworth, NJ 07033 USA Schering Plough Corp, Res Inst, Kenilworth, NJ 07033 USAZhang, Lili论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Corp, Res Inst, Kenilworth, NJ 07033 USA Schering Plough Corp, Res Inst, Kenilworth, NJ 07033 USATerracina, Giuseppe论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Corp, Res Inst, Kenilworth, NJ 07033 USA Schering Plough Corp, Res Inst, Kenilworth, NJ 07033 USA
- [10] Discovery of 3-hydroxy-4-cyano-isoquinolines as novel, potent, and selective inhibitors of human 11β-hydroxydehydrogenase 1 (11β-HSD1)BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (22) : 6693 - 6698Wu, Shung C.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAYoon, David论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAChin, Janice论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAvan Kirk, Katy论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USASeethala, Ramakrishna论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAGolla, Rajasree论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAHe, Bin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAHarrity, Thomas论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAKunselman, Lori K.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAMorgan, Nathan N.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAPonticiello, Randolph P.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USATaylor, Joseph R.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAZebo, Rachel论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAHarper, Timothy W.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USALi, Wenying论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAWang, Mengmeng论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAZhang, Lisa论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USASleczka, Bogdan G.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USANayeem, Akbar论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USASheriff, Steven论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USACamac, Daniel M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAMorin, Paul E.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAEverlof, John G.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USALi, Yi-Xin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAFerraro, Cheryl A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAKieltyka, Kasia论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAShou, Wilson论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAVath, Marianne B.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAZvyaga, Tatyana A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USAGordon, David A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USARobl, Jeffrey A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA Bristol Myers Squibb Res & Dev, Hopewell, NJ 08534 USA