Characterisation of neurokinin A induced contraction in rat and guinea-pig isolated ileum

被引：0

作者：

Maginn, M ^{[1
]}

Rea, K ^{[1
]}

Matz, J ^{[1
]}

机构：

[1] H Lundbeck A S, Dept Safety Pharmcaol, DK-2500 Copenhagen, Denmark

来源：

BRITISH JOURNAL OF PHARMACOLOGY | 2002年 / 135卷

关键词：

D O I：

暂无

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

233P

引用

页数：1

共 4 条

[1] 2(S)-((3,5-bis(trifluoromethyl)benzyl)oxy)-3(S)-phenyl-4-((3-oxo-1,2,4-triazol-5-yl)methyl)morpholine .1. A potent, orally active, morpholine-based human neurokinin-1 receptor antagonist [J].

Hale, JJ ;

Mills, SG ;

MacCoss, M ;

Shah, SK ;

Qi, HB ;

Mathre, DJ ;

Cascieri, MA ;

Sadowski, S ;

Strader, CD ;

MacIntyre, DE ;

Metzger, JM .

JOURNAL OF MEDICINAL CHEMISTRY, 1996, 39 (09) :1760-1762

[2] Tachykinin-induced contraction of the guinea-pig isolated oesophageal mucosa is mediated by NK2 receptors [J].

Kerr, KP ;

Thai, B ;

Coupar, IM .

BRITISH JOURNAL OF PHARMACOLOGY, 2000, 131 (07) :1461-1467

[3] THE NONPEPTIDE NK-2 ANTAGONIST SR 48968 IS ALSO A NK-3 ANTAGONIST IN THE GUINEA-PIG BUT NOT IN THE RAT [J].

PETITET, F ;

BEAUJOUAN, JC ;

SAFFROY, M ;

TORRENS, Y ;

GLOWINSKI, J .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1993, 191 (01) :180-187

[4] RECEPTORS FOR SUBSTANCE-P AND RELATED NEUROKININS [J].

REGOLI, D ;

DRAPEAU, G ;

DION, S ;

DORLEANSJUSTE, P .

PHARMACOLOGY, 1989, 38 (01) :1-15

← 1 →