Synthesis of optically active 1,5-benzothiazepines

被引：25

作者：

Levai, Albert ^{[1
]}

Kiss-Szikszai, Attila ^{[1
]}

机构：

[1] Univ Debrecen, Dept Organ Chem, POB 20, H-4010 Debrecen, Hungary

来源：

ARKIVOC | 2008年

关键词：

2,3-Dihydro-1,5-benzothiazepin-4(5H)-ones; 3-alkyl-2,3-dihydro-1,5-benzothiazepin4(5H)-ones; 3-amino-2,3-dihydro-1,5-benzothiazepin-4(5H)-ones; 2,3-dihydro-3-hydroxy-1,5-benzothiazepin-4(5H)-ones;

D O I：

10.3998/ark.5550190.0009.103

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Optically active 1,5-benzothiazepines belong to the well known benzothiazepine type substances. Some of them possess important bioactivities. In this review article, optically active 2,3-dihydro1,5-benzothiazepin-4(5H)-ones, their 3-amino and 3-hydroxy derivatives, comprising the most important groups of these benzothiazepines, will be discussed in detail. Less known optically active 1,5-benzothiazepines will also be included.

引用

页码：65 / 86

页数：22

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