Osimertinib as first-line treatment of EGFR mutant advanced non-small-cell lung cancer

被引:13
作者
Liam, Chong-Kin [1 ]
机构
[1] Univ Malaya, Fac Med, Dept Med, Kuala Lumpur 50603, Malaysia
关键词
SINGLE-ARM; AZD9291; MULTICENTER; RESISTANCE; MUTATIONS; ERLOTINIB; TKI;
D O I
10.21037/tlcr.2017.10.10
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:S62 / S66
页数:5
相关论文
共 18 条
[1]   The Impact of EGFR T790M Mutations and BIM mRNA Expression on Outcome in Patients with EGFR-Mutant NSCLC Treated with Erlotinib or Chemotherapy in the Randomized Phase III EURTAC Trial [J].
Costa, Carlota ;
Molina, Miguel Angel ;
Drozdowskyj, Ana ;
Gimenez-Capitan, Ana ;
Bertran-Alamillo, Jordi ;
Karachaliou, Niki ;
Gervais, Radj ;
Massuti, Bartomeu ;
Wei, Jia ;
Moran, Teresa ;
Majem, Margarita ;
Felip, Enriqueta ;
Carcereny, Enric ;
Garcia-Campelo, Rosario ;
Viteri, Santiago ;
Taron, Miquel ;
Ono, Mayumi ;
Giannikopoulos, Petros ;
Bivona, Trever ;
Rosell, Rafael .
CLINICAL CANCER RESEARCH, 2014, 20 (07) :2001-2010
[2]   AZD9291, an Irreversible EGFR TKI, Overcomes T790M-Mediated Resistance to EGFR Inhibitors in Lung Cancer [J].
Cross, Darren A. E. ;
Ashton, Susan E. ;
Ghiorghiu, Serban ;
Eberlein, Cath ;
Nebhan, Caroline A. ;
Spitzler, Paula J. ;
Orme, Jonathon P. ;
Finlay, M. Raymond V. ;
Ward, Richard A. ;
Mellor, Martine J. ;
Hughes, Gareth ;
Rahi, Amar ;
Jacobs, Vivien N. ;
Brewer, Monica Red ;
Ichihara, Eiki ;
Sun, Jing ;
Jin, Hailing ;
Ballard, Peter ;
Al-Kadhimi, Katherine ;
Rowlinson, Rachel ;
Klinowska, Teresa ;
Richmond, Graham H. P. ;
Cantarini, Mireille ;
Kim, Dong-Wan ;
Ranson, Malcolm R. ;
Pao, William .
CANCER DISCOVERY, 2014, 4 (09) :1046-1061
[3]  
Eberlein C, 2014, P AACR ANN M 2014 AP
[4]   Osimertinib for pretreated EGFR Thr790Met-positive advanced non-small-cell lung cancer (AURA2): a multicentre, open-label, single-arm, phase 2 study [J].
Goss, Glenwood ;
Tsai, Chun-Ming ;
Shepherd, Frances A. ;
Bazhenova, Lyudmila ;
Lee, Jong Seok ;
Chang, Gee-Chen ;
Crino, Lucio ;
Satouchi, Miyako ;
Chu, Quincy ;
Hida, Toyoaki ;
Han, Ji-Youn ;
Juan, Oscar ;
Dunphy, Frank ;
Nishio, Makoto ;
Kang, Jin-Hyoung ;
Majem, Margarita ;
Mann, Helen ;
Cantarini, Mireille ;
Ghiorghiu, Serban ;
Mitsudomi, Tetsuya .
LANCET ONCOLOGY, 2016, 17 (12) :1643-1652
[5]   AZD9291 in EGFR Inhibitor-Resistant Non-Small-Cell Lung Cancer [J].
Jaenne, Pasi A. ;
Yang, James Chih-Hsin ;
Kim, Dong-Wan ;
Planchard, David ;
Ohe, Yuichiro ;
Ramalingam, Suresh S. ;
Ahn, Myung-Ju ;
Kim, Sang-We ;
Su, Wu-Chou ;
Horn, Leora ;
Haggstrom, Daniel ;
Felip, Enriqueta ;
Kim, Joo-Hang ;
Frewer, Paul ;
Cantarini, Mireille ;
Brown, Kathryn H. ;
Dickinson, Paul A. ;
Ghiorghiu, Serban ;
Ranson, Malcolm .
NEW ENGLAND JOURNAL OF MEDICINE, 2015, 372 (18) :1689-1699
[6]   Osimertinib or Platinum-Pemetrexed in EGFR T790M-Positive Lung Cancer [J].
Mok, T. S. ;
Wu, Y. -L. ;
Ahn, M. -J. ;
Garassino, M. C. ;
Kim, H. R. ;
Ramalingam, S. S. ;
Shepherd, F. A. ;
He, Y. ;
Akamatsu, H. ;
Theelen, W. S. M. E. ;
Lee, C. K. ;
Sebastian, M. ;
Templeton, A. ;
Mann, H. ;
Marotti, M. ;
Ghiorghiu, S. ;
Papadimitrakopoulou, V. A. .
NEW ENGLAND JOURNAL OF MEDICINE, 2017, 376 (07) :629-640
[7]  
*NAT COMPR CANC NE, NCCN CLIN PRACT GUID
[8]   Metastatic non-small-cell lung cancer: ESMO Clinical Practice Guidelines for diagnosis, treatment and follow-up [J].
Novello, S. ;
Barlesi, F. ;
Califano, R. ;
Cufer, T. ;
Ekman, S. ;
Levra, M. Giaj ;
Kerr, K. ;
Popat, S. ;
Reck, M. ;
Senan, S. ;
Simo, G. V. ;
Vansteenkiste, J. ;
Peters, S. .
ANNALS OF ONCOLOGY, 2016, 27 :v1-v27
[9]   Association Between Plasma Genotyping and Outcomes of Treatment With Osimertinib (AZD9291) in Advanced Non-Small-Cell Lung Cancer [J].
Oxnard, Geoffrey R. ;
Thress, Kenneth S. ;
Alden, Ryan S. ;
Lawrance, Rachael ;
Paweletz, Cloud P. ;
Cantarini, Mireille ;
Yang, James Chih-Hsin ;
Barrett, J. Carl ;
Janne, Pasi A. .
JOURNAL OF CLINICAL ONCOLOGY, 2016, 34 (28) :3375-+
[10]   Acquired Resistance to EGFR Tyrosine Kinase Inhibitors in EGFR-Mutant Lung Cancer: Distinct Natural History of Patients with Tumors Harboring the T790M Mutation [J].
Oxnard, Geoffrey R. ;
Arcila, Maria E. ;
Sima, Camelia S. ;
Riely, Gregory J. ;
Chmielecki, Juliann ;
Kris, Mark G. ;
Pao, William ;
Ladanyi, Marc ;
Miller, Vincent A. .
CLINICAL CANCER RESEARCH, 2011, 17 (06) :1616-1622