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- [1] Conformation constraint of anilides enabling the discovery of tricyclic lactams as potent MK2 non-ATP competitive inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (11) : 3262 - 3266Xiao, Dong论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAPalani, Anandan论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAHuang, Xianhai论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USASofolarides, Michael论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAZhou, Wei论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAChen, Xiao论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAAslanian, Robert论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAGuo, Zhuyan论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAFossetta, James论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USATian, Fang论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USATrivedi, Prashant论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USASpacciapoli, Peter论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Kenilworth, NJ 07033 USAWhitehurst, Charles E.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Kenilworth, NJ 07033 USALundell, Daniel论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USA
- [2] Discovery and Hit-to-Lead Optimization of Non-ATP Competitive MK2 (MAPKAPK2) InhibitorsACS MEDICINAL CHEMISTRY LETTERS, 2011, 2 (08): : 632 - 637Huang, Xiaohua论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Cambridge, MA 02141 USA Merck Res Labs, Cambridge, MA 02141 USAShipps, Gerald W., Jr.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Cambridge, MA 02141 USA Merck Res Labs, Cambridge, MA 02141 USACheng, Cliff C.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Cambridge, MA 02141 USA Merck Res Labs, Cambridge, MA 02141 USASpacciapoli, Peter论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Cambridge, MA 02141 USA Merck Res Labs, Cambridge, MA 02141 USAZhang, Xingmin论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Cambridge, MA 02141 USA Merck Res Labs, Cambridge, MA 02141 USAMcCoy, Mark A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Cambridge, MA 02141 USA Merck Res Labs, Cambridge, MA 02141 USAWyss, Daniel F.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Cambridge, MA 02141 USA Merck Res Labs, Cambridge, MA 02141 USAYang, Xianshu论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Cambridge, MA 02141 USA Merck Res Labs, Cambridge, MA 02141 USAAchab, Abdelghani论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Cambridge, MA 02141 USA Merck Res Labs, Cambridge, MA 02141 USASoucy, Kyle论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Cambridge, MA 02141 USA Merck Res Labs, Cambridge, MA 02141 USAMontavon, Donna K.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Cambridge, MA 02141 USA Merck Res Labs, Cambridge, MA 02141 USAMurphy, Denise M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Cambridge, MA 02141 USA Merck Res Labs, Cambridge, MA 02141 USAWhitehurst, Charles E.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Cambridge, MA 02141 USA Merck Res Labs, Cambridge, MA 02141 USA
- [3] Discovery of a Potent Dihydrooxadiazole Series of Non-ATP-Competitive MK2 (MAPKAPK2) InhibitorsACS MEDICINAL CHEMISTRY LETTERS, 2012, 3 (02): : 100 - 105Qin, Jun论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USADhondi, Pawan论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USAHuang, Xianhai论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USAAslanian, Robert论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USAFossetta, James论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Inflammatory Dis, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USATian, Fang论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Inflammatory Dis, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USALundell, Daniel论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Inflammatory Dis, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USAPalani, Anandan论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA
- [4] Discovery of a novel series of potent MK2 non-ATP competitive inhibitors using 1,2-substituted azoles as cis-amide isosteresBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 24 (15) : 3609 - 3613Xiao, Dong论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAZhu, Xiaohong论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USASofolarides, Michael论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USADegrado, Sylvia论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAShao, Ning论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USARao, Ashwin论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAChen, Xiao论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAAslanian, Robert论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAFossetta, James论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USATian, Fang论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USATrivedi, Prashant论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USALundell, Daniel论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAPalani, Anandan论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USA
- [5] Discovery of highly potent and selective PoA MK2 inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 248Mogemark, Mickael T.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Med Chem, Molndal, Sweden AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Med Chem, Molndal, SwedenEvertsson, Emma论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Med Chem, Molndal, Sweden AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Med Chem, Molndal, Swedenaf Rosenschold, Magnus Munck论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Med Chem, Molndal, Sweden AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Med Chem, Molndal, SwedenNorberg, Monica论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Med Chem, Molndal, Sweden AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Med Chem, Molndal, SwedenLever, Sarah论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Med Chem, Molndal, Sweden AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Med Chem, Molndal, SwedenLonn, Hans论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Med Chem, Molndal, Sweden AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Med Chem, Molndal, SwedenPardali, Katerina论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Translat Sci, Molndal, Sweden AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Med Chem, Molndal, SwedenHedstrom, Ulf论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Translat Sci, Molndal, Sweden AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Med Chem, Molndal, SwedenBold, Peter论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept DMPK, Molndal, Sweden AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Med Chem, Molndal, SwedenDavis, Andy论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Biosci, Molndal, Sweden AstraZeneca R&D, Resp Inflammat & Autoimmun iMed, Dept Med Chem, Molndal, Sweden
- [6] Computational Insights for the Discovery of Non-ATP Competitive Inhibitors of MAP KinasesCURRENT PHARMACEUTICAL DESIGN, 2012, 18 (09) : 1173 - 1185Schnieders, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Austin, Dept Biomed Engn, Austin, TX 78712 USA Univ Texas Austin, Dept Biomed Engn, Austin, TX 78712 USAKaoud, Tamer S.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Austin, Div Med Chem, Austin, TX 78712 USA Univ Texas Austin, Grad Programs Pharm, Austin, TX 78712 USA Univ Texas Austin, Dept Biomed Engn, Austin, TX 78712 USAYan, Chunli论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Austin, Dept Biomed Engn, Austin, TX 78712 USA Univ Texas Austin, Dept Biomed Engn, Austin, TX 78712 USADalby, Kevin N.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Austin, Div Med Chem, Austin, TX 78712 USA Univ Texas Austin, Grad Programs Biochem, Austin, TX 78712 USA Univ Texas Austin, Dept Biomed Engn, Austin, TX 78712 USARen, Pengyu论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Austin, Dept Biomed Engn, Austin, TX 78712 USA Univ Texas Austin, Grad Programs Biomed Engn, Austin, TX 78712 USA Univ Texas Austin, Dept Biomed Engn, Austin, TX 78712 USA
- [7] Non-ATP Competitive Protein Kinase InhibitorsCURRENT MEDICINAL CHEMISTRY, 2010, 17 (25) : 2804 - 2821Garuti, L.论文数: 0 引用数: 0 h-index: 0机构: Univ Bologna, Dept Pharmaceut Sci, I-40126 Bologna, Italy Univ Bologna, Dept Pharmaceut Sci, I-40126 Bologna, ItalyRoberti, M.论文数: 0 引用数: 0 h-index: 0机构: Univ Bologna, Dept Pharmaceut Sci, I-40126 Bologna, Italy Univ Bologna, Dept Pharmaceut Sci, I-40126 Bologna, ItalyBottegoni, G.论文数: 0 引用数: 0 h-index: 0机构: Italian Inst Technol, Dept Drug Discovery & Dev, I-16163 Genoa, Italy Univ Bologna, Dept Pharmaceut Sci, I-40126 Bologna, Italy
- [8] Novel ATP competitive MK2 inhibitors with potent biochemical and cell-based activity throughout the seriesBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (01) : 613 - 618Oubrie, Arthur论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsKaptein, Allard论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, Netherlandsde Zwart, Edwin论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsHoogenboom, Niels论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsGoorden, Rianne论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, Netherlandsvan de Kar, Bas论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, Netherlandsvan Hoek, Maaike论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, Netherlandsde Kimpe, Vera论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, Netherlandsvan der Heijden, Ruud论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsBorsboom, Judith论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsKazemier, Bert论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, Netherlandsde Roos, Jeroen论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsScheffers, Michiel论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsLommerse, Jos论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsSchultz-Fademrecht, Carsten论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsBarf, Tjeerd论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands
- [9] Discovery of selective and orally available spiro-3-piperidyl ATP-competitive MK2 inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (12) : 3823 - 3827Kaptein, Allard论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsOubrie, Arthur论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, Netherlandsde Zwart, Edwin论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsHoogenboom, Niels论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, Netherlandsde Wit, Joeri论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, Netherlandsvan de Kar, Bas论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, Netherlandsvan Hoek, Maaike论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsVogel, Gerard论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, Netherlandsde Kimpe, Vera论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsSchultz-Fademrecht, Carsten论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsBorsboom, Judith论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, Netherlandsvan Zeeland, Mario论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsVersteegh, Judith论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsKazemier, Bert论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, Netherlandsde Roos, Jeroen论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsWijnands, Frank论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsDulos, John论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsJaeger, Martin论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsLeandro-Garcia, Paula论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, NetherlandsBarf, Tjeerd论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands Merck Res Labs, MSD, NL-5340 BH Oss, Netherlands
- [10] Discovery of the first non-ATP competitive IGF-1R kinase inhibitors: Advantages in comparison with competitive inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (08) : 2224 - 2228Lesuisse, Dominique论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Med Chem, F-94300 Vitry Sur Seine, France Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USAMauger, Jacques论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USA Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USANemecek, Conception论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Med Chem, F-94300 Vitry Sur Seine, France Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USAMaignan, Sebastien论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Struct Biol & Mol Modelling, F-94300 Vitry Sur Seine, France Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USABoiziau, Janine论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Oncol Therapeut Domain, F-94300 Vitry Sur Seine, France Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USAHarlow, Greg论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USA Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USAHittinger, Augustin论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Med Chem, F-94300 Vitry Sur Seine, France Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USARuf, Swen论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Med Chem, D-65926 Frankfurt, Germany Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USAStrobel, Hartmut论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Med Chem, D-65926 Frankfurt, Germany Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USANair, Anil论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USA Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USARitter, Kurt论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Med Chem, D-65926 Frankfurt, Germany Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USAMalleron, Jean-Luc论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Med Chem, F-94300 Vitry Sur Seine, France Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USADagallier, Anne论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Struct Biol & Mol Modelling, F-94300 Vitry Sur Seine, France Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USAEl-Ahmad, Youssef论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Med Chem, F-94300 Vitry Sur Seine, France Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USAGuilloteau, Jean-Pierre论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Struct Biol & Mol Modelling, F-94300 Vitry Sur Seine, France Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USAGuizani, Houlfa论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Med Chem, F-94300 Vitry Sur Seine, France Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USABouchard, Herve论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Med Chem, F-94300 Vitry Sur Seine, France Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USAVenot, Corinne论文数: 0 引用数: 0 h-index: 0机构: Sanofi Aventis, Oncol Therapeut Domain, F-94300 Vitry Sur Seine, France Sanofi Aventis, Highthroughput Med Chem, Oro Valle, AZ 85755 USA