Solubility of mesalazine in polyethylene glycol 400+water mixtures at different temperatures

被引：15
作者：
Moradi, Milad [1 ,2 ,3 ]
Rahimpour, Elaheh [2 ,3 ,4 ]
Hemmati, Salar [5 ]
Martinez, Fleming [6 ]
Barzegar-Jalali, Mohammad [3 ,7 ]
Jouyban, Abolghasem [2 ,3 ,8 ]
机构：
[1] Tabriz Univ Med Sci, Fac Pharm, Student Res Comm, Tabriz, Iran
[2] Tabriz Univ Med Sci, Pharmaceut Anal Res Ctr, Tabriz, Iran
[3] Tabriz Univ Med Sci, Fac Pharm, Tabriz, Iran
[4] Tabriz Univ Med Sci, Food & Drug Safety Res Ctr, Tabriz, Iran
[5] Tabriz Univ Med Sci, Drug Appl Res Ctr, Tabriz, Iran
[6] Univ Nacl Colombia, Fac Ciencias, Dept Farm, Grp Invest Farmaceut Fisicoquim,Sede Bogota, Cra 30 45-03, Bogota, DC, Colombia
[7] Tabriz Univ Med Sci, Res Ctr Pharmaceut Nanotechnol, Tabriz, Iran
[8] Univ Tehran Med Sci, Digest Dis Res Inst, Tehran, Iran
来源：
JOURNAL OF MOLECULAR LIQUIDS | 2020年 / 314卷
关键词：
Solubility; Mesalazine; Polyethylene glycol 400; Cosolvency models; Dissolution thermodynamics; Preferential solvation; PREFERENTIAL SOLVATION; COSOLVENCY; PREDICTION; MODELS; DRUGS;
D O I：
10.1016/j.molliq.2020.113546
中图分类号：
O64 [物理化学（理论化学）、化学物理学];
学科分类号：
070304 ; 081704 ;
摘要：
Temperature-dependent solubility data for mesalazine in the binary system of polyethylene glycol 400 (PEG 400)/water are determined by a shake-flask method at 293.2-313.2 K. The solubility data are validated to five different computational models including the van't Hoff, the mixture response surface, the Yalkowsky, the Jouyban-Acree, and the Jouyban-Acree-van't Hoff. All the investigated models have good correlation and validation according to obtained the mean relative deviations (MRD%) for back-calculated data. Moreover, apparent thermodynamic analysis shows an endothemiic process for mesalazine in (PEG 400 +/- water) mixtures. Further, based on inverse Kirkwood-Buff integrals is observed that mesalazine is preferentially solvated by PEG in all the mixtures. (C) 2020 Elsevier B.V. All rights reserved.
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页数：8
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