A facile synthesis of various fluorine-containing indole derivatives via palladium-catalyzed annulation of internal alkynes

被引：46

作者：

Chae, J ^{[1
]}

Konno, T ^{[1
]}

Ishihara, T ^{[1
]}

Yamanaka, H ^{[1
]}

机构：

[1] Kyoto Inst Technol, Dept Chem & Mat Technol, Sakyo Ku, Kyoto 6068585, Japan

来源：

CHEMISTRY LETTERS | 2004年 / 33卷 / 03期

关键词：

D O I：

10.1246/cl.2004.314

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

The palladium-catalyzed annulation reaction of a variety of fluorine-containing internal alkynes with 2-iodoaniline derivatives took place smoothly to give the corresponding 2,3-disubstituted indole derivatives in good to excellent yields.

引用

页码：314 / 315

页数：2

共 14 条

[11] SYNTHETICALLY ATTRACTIVE INDOLIZATION PROCESSES AND NEWER METHODS FOR THE PREPARATION OF SELECTIVELY SUBSTITUTED INDOLES [J].

PINDUR, U ;

ADAM, R .

JOURNAL OF HETEROCYCLIC CHEMISTRY, 1988, 25 (01) :1-8

[12] PERFLUOROPROPYLATION OF FURANS, THIOPHENES, AND PYRIDINES WITH BIS(HEPTAFLUOROBUTYRYL) PEROXIDE [J].

SAWADA, H ;

YOSHIDA, M ;

HAGII, H ;

AOSHIMA, K ;

KOBAYASHI, M .

BULLETIN OF THE CHEMICAL SOCIETY OF JAPAN, 1986, 59 (01) :215-219

[13] ADVANCES IN THE PREPARATION OF BIOLOGICALLY-ACTIVE ORGANOFLUORINE COMPOUNDS [J].

WELCH, JT .

TETRAHEDRON, 1987, 43 (14) :3123-3197

[14] PERFLUOROALKYLATIONS OF NITROGEN-CONTAINING HETEROAROMATIC-COMPOUNDS WITH BIS(PERFLUOROALKANOYL) PEROXIDES [J].

YOSHIDA, M ;

YOSHIDA, T ;

KOBAYASHI, M ;

KAMIGATA, N .

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1989, (05) :909-914

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