Facile synthesis of some novel 1,3,4,2-oxa(thia)diazaphospholo[5,4-b]quinazolinones and 1,2,4,3-triazaphospholo[5,1-b]quinazolinones

被引：4

作者：

Ali, Tarik E. ^{[1
,2
]}

Assiri, Mohammed A. ^{[1
]}

Zahran, H. Y. ^{[3
,4
,5
]}

Yahia, I. S. ^{[3
,4
,5
]}

Hussien, Mai S. A. ^{[2
]}

机构：

[1] King Khalid Univ, Fac Sci, Dept Chem, Abha, Saudi Arabia

[2] Ain Shams Univ, Fac Educ, Dept Chem, Cairo, Egypt

[3] King Khalid Univ, Res Ctr Adv Mat Sci, Abha, Saudi Arabia

[4] King Khalid Univ, Fac Sci, Dept Phys, Abha, Saudi Arabia

[5] Ain Shams Univ, Fac Educ, Dept Phys, Cairo, Egypt

来源：

SYNTHETIC COMMUNICATIONS | 2021年 / 51卷 / 02期

关键词：

Cyclocondensation; 1; 3; 4; 2-oxadiazaphosphole; quinazolinone; 2-thiadiazaphosphole; 2; 3-triazaphosphole; FUSED HETEROCYCLES; DESIGN; DERIVATIVES;

D O I：

10.1080/00397911.2020.1825745

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The cyclo condensation of some bi-functionally quinazolinones with some phosphorus dihalides in dry pyridine led to novel 1,3,4,2-oxadiazaphospholo[5,4-b]quinazolinones, 1,3,4,2-thiadiazaphospholo[5,4-b]quinazolinones and 1,2,4,3-triazaphospholo[5,1-b]quinazolinones. The structure of novel products was established by IR and NMR spectroscopy.

引用

页码：302 / 307

页数：6

共 29 条

[1] Abd El-Dayem NS., 2020, J APPL CHEM-USSR, V13, P49, DOI DOI 10.9790/5736-1302014964
[2] Design, synthesis of 2,3-disubstitued 4(3H)-quinazolinone derivatives as anti-inflammatory and analgesic agents: COX-1/2 inhibitory activities and molecular docking studies
Abdel-Aziz, Alaa A. -M.
Abou-Zeid, Laila A.
ElTahir, Kamal Eldin H.
Mohamed, Menshawy A.
Abu El-Enin, Mohamed A.
El-Azab, Adel S.
[J]. BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 24 (16) : 3818 - 3828
[3] ABDELALIM AAM, 1994, INDIAN J CHEM B, V33, P260
[4] Synthesis of [1,5-c]quinazolo-1,2,4,3-triazaphosphole 4-oxide
Abderrahim, R
Boujlel, K
[J]. PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS, 2005, 180 (01) : 79 - 84
[5] Convenient synthesis of [1,5-c]quinazolo-2,3-dihydro-1,2,4,3-triazaphospholes and [1,5-c]quinazolo-2,3-dihydro-1,2,4,3-triazaphosphole-3-sulfides
Abderrahim, Raoudha
[J]. PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS, 2007, 182 (04) : 893 - 897
[6] Use of phosphonyl carbanions in the synthesis of anti-inflammatory active phosphorus-containing fused heterocycles and relevance phosphonates
Abdou, Wafaa M.
Kamel, Azza A.
Shaddy, Abeer A.
[J]. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2010, 45 (11) : 5217 - 5224
[7] Synthesis and antihypertensive activity of novel 3-benzyl-2-substituted-3H-[1,2,4]triazolo[5,1-b]quinazolin-9-ones
Alagarsamy, Veerachamy
Pathak, Urvishbhai S.
[J]. BIOORGANIC & MEDICINAL CHEMISTRY, 2007, 15 (10) : 3457 - 3462
[8] FIRST SYNTHESIS OF BENZO [e] [1,3,2]DIAZAPHOSPHININO[1,6-c]-[1,3,2]OXAZAPHOSPHININES
Ali, Tarik E.
Assiri, Mohammed A.
Yahia, Ibrahim S.
[J]. HETEROCYCLES, 2019, 98 (09) : 1265 - 1272
[9] Facile synthesis of novel 6-methyl-5-phenyl-2-sulfido-1,2,3,5-tetrahydro-4H[1,2] oxazolo[4′,5′:5,6]pyrano[2,3-d][1,3,2] diazaphosphinines
Ali, Tarik E.
Assiri, Mohamed A.
Abdel-Kariem, Somaia M.
Yahia, Ibrahim S.
[J]. JOURNAL OF SULFUR CHEMISTRY, 2018, 39 (05) : 472 - 482
[10] Reaction of 2-cyano-3-(4-oxo-4H-chromen-3-yl)prop-2-enamide with some phosphorus reagents: synthesis of some novel diethyl phosphonates, 1,2,3-diazaphosphinanes, 1,2,3-thiazaphosphinine and 1,2-azaphospholes bearing a chromone ring
Ali, Tarik E.
Hassan, Mohamed M.
[J]. RESEARCH ON CHEMICAL INTERMEDIATES, 2018, 44 (01) : 173 - 189

← 1 2 3 →