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- [1] MEDI 404-SAR studies on a novel series of potent ACC2 inhibitors for treatment of obesity and type 2 diabetesABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2006, 232Zhang, Tianyuan论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Abbott Pk, IL 66064 USA Abbott Labs, Abbott Pk, IL 66064 USAClark, Richard F.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R4CV, Abbott Pk, IL 60064 USA Abbott Labs, Abbott Pk, IL 66064 USAHansen, Todd M.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Abbott Pk, IL 66064 USA Abbott Labs, Abbott Pk, IL 66064 USAXin, Zhili论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Abbott Pk, IL 66064 USALiu, Gang论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Abbott Pk, IL 66064 USAWang, Xiaojun论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Abbott Pk, IL 66064 USA Abbott Labs, Abbott Pk, IL 66064 USAWang, Rongqi论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Abbott Pk, IL 66064 USA Abbott Labs, Abbott Pk, IL 66064 USACamp, Heidi S.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res Div, Abbott Pk, IL 60064 USA Abbott Labs, Abbott Pk, IL 66064 USABeutel, Bruce A.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept 47P, Abbott Pk, IL 60064 USA Abbott Labs, Abbott Pk, IL 66064 USASham, Hing论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, GPRD, Abbott Pk, IL 60064 USA Abbott Labs, Abbott Pk, IL 66064 USAGu, Yu Gui论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Abbott Pk, IL 66064 USA Abbott Labs, Abbott Pk, IL 66064 USA
- [2] Discovery of a Novel 2,6-Disubstituted Glucosamine Series of Potent and Selective Hexokinase 2 InhibitorsACS MEDICINAL CHEMISTRY LETTERS, 2016, 7 (03): : 217 - 222Lin, Hong论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USAZeng, Jin论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USAXie, Ren论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USASchulz, Mark J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USATedesco, Rosanna论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USAQu, Junya论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USAErhard, Karl F.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USAMack, James F.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USARaha, Kaushik论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USARendina, Alan R.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USASzewczuk, Lawrence M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USAKratz, Patricia M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USAJurewicz, Anthony J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USACecconie, Ted论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USAMartens, Stan论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USAMcDevit, Patrick J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USAMartin, John D.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USAChen, Stephenie B.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USAJiang, Yong论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USANickels, Leng论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USASchwartz, Benjamin J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USASmallwood, Angela论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USAZhao, Baoguang论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USACampobasso, Nino论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USAQian, Yanqiu论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USABriand, Jacques论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USARominger, Cynthia M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Metab Biol, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USAOleykowski, Catherine论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Metab Biol, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USAHardwicke, Mary Ann论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Metab Biol, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USALuengo, Juan I.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Metab Chem, 1250 South Collegeville Rd, Collegeville, PA 19426 USA
- [3] Discovery and Biological Evaluation of a Novel Highly Potent Selective Butyrylcholinsterase InhibitorJOURNAL OF MEDICINAL CHEMISTRY, 2020, 63 (17) : 10030 - 10044Li, Qi论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaXing, Shuaishuai论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaChen, Ying论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Dept Nat Med Chem, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaLiao, Qinghong论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Dept Nat Med Chem, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaXiong, Baichen论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Dept Nat Med Chem, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaHe, Siyu论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Jiangsu Key Lab Carcinogenesis & Intervent, Sch Basic Med & Clin Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaLu, Weixuan论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaLiu, Yang论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaYang, Hongyu论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaLi, Qihang论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaFeng, Feng论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Dept Nat Med Chem, Nanjing 211198, Peoples R China Jiangsu Food & Pharmaceut Sci Coll, Huaian 223003, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaLiu, Wenyuan论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaChen, Yao论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaSun, Haopeng论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China
- [4] Discovery of Potent and Selective RSK Inhibitors as Biological ProbesJOURNAL OF MEDICINAL CHEMISTRY, 2015, 58 (17) : 6766 - 6783Jain, Rama论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USAMathur, Michelle论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USALan, Jiong论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USACostales, Abran论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USAAtallah, Gordana论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USARamurthy, Savithri论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USASubramanian, Sharadha论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USASetti, Lina论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USAFeucht, Paul论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USAWarne, Bob论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USADoyle, Laura论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USABasham, Stephen论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USAJefferson, Anne B.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USALindvall, Mika论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USAAppleton, Brent A.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USAShafer, Cynthia M.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Global Discovery Chem Oncol & Exploratory Chem, Emeryville, CA 94608 USA
- [5] A novel series of potent and selective IKK2 inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2004, 14 (02) : 409 - 412Bingham, AH论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Cambridge CB1 6GS, England Celltech R&D Ltd, Cambridge CB1 6GS, EnglandDavenport, RJ论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Cambridge CB1 6GS, England Celltech R&D Ltd, Cambridge CB1 6GS, EnglandGowers, L论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Cambridge CB1 6GS, England Celltech R&D Ltd, Cambridge CB1 6GS, EnglandKnight, RL论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Cambridge CB1 6GS, England Celltech R&D Ltd, Cambridge CB1 6GS, EnglandLowe, C论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Cambridge CB1 6GS, England Celltech R&D Ltd, Cambridge CB1 6GS, EnglandOwen, DA论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Cambridge CB1 6GS, England Celltech R&D Ltd, Cambridge CB1 6GS, EnglandParry, DM论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Cambridge CB1 6GS, England Celltech R&D Ltd, Cambridge CB1 6GS, EnglandPitt, WR论文数: 0 引用数: 0 h-index: 0机构: Celltech R&D Ltd, Cambridge CB1 6GS, England Celltech R&D Ltd, Cambridge CB1 6GS, England
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