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- [1] BRD4 Degradation By Protacs Represents a More Effective Therapeutic Strategy Than BRD4 Inhibitors in DLBCLBLOOD, 2015, 126 (23)Lu, Jing论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, New Haven, CT USA Arvinas LLC, New Haven, CT USAQian, Yimin论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, New Haven, CT USA Arvinas LLC, New Haven, CT USARaina, Kanak论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, New Haven, CT USA Arvinas LLC, New Haven, CT USAAltieri, Martha论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, New Haven, CT USA Arvinas LLC, New Haven, CT USADong, Hanqing论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, New Haven, CT USA Arvinas LLC, New Haven, CT USAWang, Jing论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, New Haven, CT USA Arvinas LLC, New Haven, CT USAChen, Xin论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, New Haven, CT USA Arvinas LLC, New Haven, CT USACrew, Andrew论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, New Haven, CT USA Arvinas LLC, New Haven, CT USAColeman, Kevin论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, New Haven, CT USA Arvinas LLC, New Haven, CT USACrews, Craig论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Dept Mol Cellular & Dev Biol, Dept Chem, Dept Pharmacol, New Haven, CT USA Arvinas LLC, New Haven, CT USAWinkler, James论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, New Haven, CT USA Arvinas LLC, New Haven, CT USA
- [2] Methylation of BRD4 by PRMT1 regulates BRD4 phosphorylation and promotes ovarian cancer invasionCELL DEATH & DISEASE, 2023, 14 (09)Liu, Yi论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R China Harvard Med Sch, Beth Israel Deaconess Med Ctr, Dept Pathol, Boston, MA 02115 USA Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R ChinaLiu, Hejing论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R China Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R ChinaYe, Miaomiao论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R China Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R ChinaJiang, Mengying论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R China Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R ChinaChen, Xin论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R China Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R ChinaSong, Gendi论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R China Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R ChinaJi, Huihui论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R China Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R ChinaWang, Zhi-wei论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R China Harvard Med Sch, Beth Israel Deaconess Med Ctr, Dept Pathol, Boston, MA 02115 USA Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R ChinaZhu, Xueqiong论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R China Wenzhou Med Univ, Dept Obstet & Gynecol, Zhejiang Prov Clin Res Ctr Obstet & Gynecol, Affiliated Hosp 2, Wenzhou 325027, Peoples R China
- [3] Methylation of BRD4 by PRMT1 regulates BRD4 phosphorylation and promotes ovarian cancer invasionCell Death & Disease, 14Yi Liu论文数: 0 引用数: 0 h-index: 0机构: the Second Affiliated Hospital of Wenzhou Medical University,Zhejiang Provincial Clinical Research Center for Obstetrics and Gynecology, Department of Obstetrics and GynecologyHejing Liu论文数: 0 引用数: 0 h-index: 0机构: the Second Affiliated Hospital of Wenzhou Medical University,Zhejiang Provincial Clinical Research Center for Obstetrics and Gynecology, Department of Obstetrics and GynecologyMiaomiao Ye论文数: 0 引用数: 0 h-index: 0机构: the Second Affiliated Hospital of Wenzhou Medical University,Zhejiang Provincial Clinical Research Center for Obstetrics and Gynecology, Department of Obstetrics and GynecologyMengying Jiang论文数: 0 引用数: 0 h-index: 0机构: the Second Affiliated Hospital of Wenzhou Medical University,Zhejiang Provincial Clinical Research Center for Obstetrics and Gynecology, Department of Obstetrics and GynecologyXin Chen论文数: 0 引用数: 0 h-index: 0机构: the Second Affiliated Hospital of Wenzhou Medical University,Zhejiang Provincial Clinical Research Center for Obstetrics and Gynecology, Department of Obstetrics and GynecologyGendi Song论文数: 0 引用数: 0 h-index: 0机构: the Second Affiliated Hospital of Wenzhou Medical University,Zhejiang Provincial Clinical Research Center for Obstetrics and Gynecology, Department of Obstetrics and GynecologyHuihui Ji论文数: 0 引用数: 0 h-index: 0机构: the Second Affiliated Hospital of Wenzhou Medical University,Zhejiang Provincial Clinical Research Center for Obstetrics and Gynecology, Department of Obstetrics and GynecologyZhi-wei Wang论文数: 0 引用数: 0 h-index: 0机构: the Second Affiliated Hospital of Wenzhou Medical University,Zhejiang Provincial Clinical Research Center for Obstetrics and Gynecology, Department of Obstetrics and GynecologyXueqiong Zhu论文数: 0 引用数: 0 h-index: 0机构: the Second Affiliated Hospital of Wenzhou Medical University,Zhejiang Provincial Clinical Research Center for Obstetrics and Gynecology, Department of Obstetrics and Gynecology
- [4] Targeting Brd4 for cancer therapy: inhibitors and degradersMEDCHEMCOMM, 2018, 9 (11) : 1779 - 1802Duan, Yingchao论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaGuan, Yuanyuan论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaQin, Wenping论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaZhai, Xiaoyu论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaYu, Bin论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Key Lab Adv Pharmaceut Technol,Sch Pharmaceutical, Minist Educ China,Inst Drug Discovery & Dev, Coinnovat Ctr Henan Prov New Drug R&D Preclin Saf, Zhengzhou 450001, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaLiu, Hongmin论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Key Lab Adv Pharmaceut Technol,Sch Pharmaceutical, Minist Educ China,Inst Drug Discovery & Dev, Coinnovat Ctr Henan Prov New Drug R&D Preclin Saf, Zhengzhou 450001, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China
- [5] Dual HDAC/BRD4 inhibitors against cancerMEDICINAL CHEMISTRY RESEARCH, 2021, 30 (10) : 1822 - 1836Omidkhah, Negar论文数: 0 引用数: 0 h-index: 0机构: Mashhad Univ Med Sci, Pharmaceut Technol Inst, Biotechnol Res Ctr, Mashhad, Iran Mashhad Univ Med Sci, Sch Pharm, Dept Med Chem, Mashhad, Iran Mashhad Univ Med Sci, Pharmaceut Technol Inst, Biotechnol Res Ctr, Mashhad, IranHadizadeh, Farzin论文数: 0 引用数: 0 h-index: 0机构: Mashhad Univ Med Sci, Pharmaceut Technol Inst, Biotechnol Res Ctr, Mashhad, Iran Mashhad Univ Med Sci, Sch Pharm, Dept Med Chem, Mashhad, Iran Mashhad Univ Med Sci, Pharmaceut Technol Inst, Biotechnol Res Ctr, Mashhad, IranGhodsi, Razieh论文数: 0 引用数: 0 h-index: 0机构: Mashhad Univ Med Sci, Pharmaceut Technol Inst, Biotechnol Res Ctr, Mashhad, Iran Mashhad Univ Med Sci, Sch Pharm, Dept Med Chem, Mashhad, Iran Mashhad Univ Med Sci, Pharmaceut Technol Inst, Biotechnol Res Ctr, Mashhad, Iran
- [6] Dual HDAC/BRD4 inhibitors against cancerMedicinal Chemistry Research, 2021, 30 : 1822 - 1836Negar Omidkhah论文数: 0 引用数: 0 h-index: 0机构: Mashhad University of Medical Sciences,Biotechnology Research Center, Pharmaceutical Technology InstituteFarzin Hadizadeh论文数: 0 引用数: 0 h-index: 0机构: Mashhad University of Medical Sciences,Biotechnology Research Center, Pharmaceutical Technology InstituteRazieh Ghodsi论文数: 0 引用数: 0 h-index: 0机构: Mashhad University of Medical Sciences,Biotechnology Research Center, Pharmaceutical Technology Institute
- [7] BRD4 inhibitors block telomere elongationNUCLEIC ACIDS RESEARCH, 2017, 45 (14) : 8403 - 8410Wang, Steven论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Univ, Sch Med, Dept Mol Biol & Genet, Baltimore, MD 21205 USA Johns Hopkins Univ, Sch Med, Cellular & Mol Med Grad Program, Baltimore, MD 21205 USA Johns Hopkins Univ, Sch Med, Dept Mol Biol & Genet, Baltimore, MD 21205 USAPike, Alexandra M.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Univ, Sch Med, Dept Mol Biol & Genet, Baltimore, MD 21205 USA Johns Hopkins Univ, Sch Med, Cellular & Mol Med Grad Program, Baltimore, MD 21205 USA Johns Hopkins Univ, Sch Med, Dept Mol Biol & Genet, Baltimore, MD 21205 USALee, Stella S.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Univ, Sch Med, Dept Mol Biol & Genet, Baltimore, MD 21205 USA US FDA, Off Commissioner, Silver Spring, MD 20993 USA Johns Hopkins Univ, Sch Med, Dept Mol Biol & Genet, Baltimore, MD 21205 USAStrong, Margaret A.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Univ, Sch Med, Dept Mol Biol & Genet, Baltimore, MD 21205 USA Johns Hopkins Univ, Sch Med, Dept Mol Biol & Genet, Baltimore, MD 21205 USAConnelly, Carla J.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Univ, Sch Med, Dept Mol Biol & Genet, Baltimore, MD 21205 USA Johns Hopkins Univ, Sch Med, Dept Mol Biol & Genet, Baltimore, MD 21205 USAGreider, Carol W.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Univ, Sch Med, Dept Mol Biol & Genet, Baltimore, MD 21205 USA Johns Hopkins Univ, Sch Med, Dept Mol Biol & Genet, Baltimore, MD 21205 USA
- [8] Review on: BRD4 inhibitors for anticancer researchHUMAN GENE, 2023, 37Singh, Vindhya Vikram论文数: 0 引用数: 0 h-index: 0机构: Shibli Natl Coll, Dept Chem, Cheminformat & Mol Modelling Lab, Azamgarh 276001, Uttar Pradesh, India Shibli Natl Coll, Dept Chem, Cheminformat & Mol Modelling Lab, Azamgarh 276001, Uttar Pradesh, IndiaAlauddin, Shafqat论文数: 0 引用数: 0 h-index: 0机构: Shibli Natl Coll, Dept Chem, Cheminformat & Mol Modelling Lab, Azamgarh 276001, Uttar Pradesh, India Shibli Natl Coll, Dept Chem, Cheminformat & Mol Modelling Lab, Azamgarh 276001, Uttar Pradesh, India
- [9] Adjusted degradation of BRD4 S and BRD4 L based on fine structural modifications of the pyrrolopyridone scaffoldEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 236Chen, Jingjing论文数: 0 引用数: 0 h-index: 0机构: UCAS, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, 1 Xiangshanzhi Rd, Hangzhou 310024, Peoples R China UCAS, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, 1 Xiangshanzhi Rd, Hangzhou 310024, Peoples R ChinaHe, Huixin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19 Yuquan Rd, Beijing 110039, Peoples R China UCAS, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, 1 Xiangshanzhi Rd, Hangzhou 310024, Peoples R ChinaWei, Aihuan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R China UCAS, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, 1 Xiangshanzhi Rd, Hangzhou 310024, Peoples R ChinaLi, Yalei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China UCAS, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, 1 Xiangshanzhi Rd, Hangzhou 310024, Peoples R ChinaCheng, Gang论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Chinese Med Univ, Coll Pharmaceut Sci, 548 Binwen Rd, Hangzhou 310053, Peoples R China UCAS, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, 1 Xiangshanzhi Rd, Hangzhou 310024, Peoples R ChinaQin, Hui论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19 Yuquan Rd, Beijing 110039, Peoples R China UCAS, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, 1 Xiangshanzhi Rd, Hangzhou 310024, Peoples R ChinaZhong, Hanyue论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19 Yuquan Rd, Beijing 110039, Peoples R China UCAS, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, 1 Xiangshanzhi Rd, Hangzhou 310024, Peoples R ChinaLiu, Hongchun论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China UCAS, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, 1 Xiangshanzhi Rd, Hangzhou 310024, Peoples R ChinaGeng, Meiyu论文数: 0 引用数: 0 h-index: 0机构: UCAS, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, 1 Xiangshanzhi Rd, Hangzhou 310024, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19 Yuquan Rd, Beijing 110039, Peoples R China UCAS, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, 1 Xiangshanzhi Rd, Hangzhou 310024, Peoples R ChinaShen, Aijun论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19 Yuquan Rd, Beijing 110039, Peoples R China UCAS, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, 1 Xiangshanzhi Rd, Hangzhou 310024, Peoples R ChinaHu, Youhong论文数: 0 引用数: 0 h-index: 0机构: UCAS, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, 1 Xiangshanzhi Rd, Hangzhou 310024, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19 Yuquan Rd, Beijing 110039, Peoples R China UCAS, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, 1 Xiangshanzhi Rd, Hangzhou 310024, Peoples R China
- [10] BRD4 is a new therapeutic target in melanomaCANCER RESEARCH, 2013, 73Fontanals-Cirera, Barbara论文数: 0 引用数: 0 h-index: 0机构: NYU, Sch Med, New York, NY USA NYU, Sch Med, New York, NY USASegura, Miguel F.论文数: 0 引用数: 0 h-index: 0机构: Vall Hebron Inst Recerca, Barcelona, Spain NYU, Sch Med, New York, NY USAGaziel-Sovran, Avital论文数: 0 引用数: 0 h-index: 0机构: NYU, Sch Med, New York, NY USA NYU, Sch Med, New York, NY USAGuijarro, Maria V.论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Gainesville, FL USA NYU, Sch Med, New York, NY USAHanniford, Doug论文数: 0 引用数: 0 h-index: 0机构: NYU, Sch Med, New York, NY USA NYU, Sch Med, New York, NY USAGonzalez-Gomez, Pilar论文数: 0 引用数: 0 h-index: 0机构: Inst Salud Carlos III, Madrid, Spain NYU, Sch Med, New York, NY USAZhang, Weijia论文数: 0 引用数: 0 h-index: 0机构: Mt Sinai Sch Med, New York, NY USA NYU, Sch Med, New York, NY USAZhang, Guantao论文数: 0 引用数: 0 h-index: 0机构: Mt Sinai Sch Med, New York, NY USA NYU, Sch Med, New York, NY USADarvishian, Farbod论文数: 0 引用数: 0 h-index: 0机构: NYU, Sch Med, New York, NY USA NYU, Sch Med, New York, NY USAOhlmeyer, Michael论文数: 0 引用数: 0 h-index: 0机构: Mt Sinai Sch Med, New York, NY USA NYU, Sch Med, New York, NY USAOsman, Iman论文数: 0 引用数: 0 h-index: 0机构: NYU, Sch Med, New York, NY USA NYU, Sch Med, New York, NY USAZhou, Ming-Ming论文数: 0 引用数: 0 h-index: 0机构: Mt Sinai Sch Med, New York, NY USA NYU, Sch Med, New York, NY USAHernando, Eva论文数: 0 引用数: 0 h-index: 0机构: NYU, Sch Med, New York, NY USA NYU, Sch Med, New York, NY USA