Palladium heteroannulation process for synthesis of substituted pyrrolo [2,3-b]pyridin-3-ones

被引：51

作者：

Desarbre, E ^{[1
]}

Merour, JY ^{[1
]}

机构：

[1] UNIV ORLEANS,CNRS,INST CHIM ORGAN & ANALYT,F-45067 ORLEANS 2,FRANCE

来源：

TETRAHEDRON LETTERS | 1996年 / 37卷 / 01期

关键词：

D O I：

10.1016/0040-4039(95)02079-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Substituted-3H-pyrrolo[2,3-b]pyridin-3-ones 7b-d were prepared from 2-amino-3-iodopyridine derivatives 3b-d by palladium carboannulation process with allenic compounds and then oxidative cleavage of the exocyclic carbon-carbon double bond.

引用

页码：43 / 46

页数：4

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