Dienediolates of α,β-unsaturated carboxylic acids in synthesis:: A new synthetic method to 2-pyridones

被引：0

作者：

Brun, EM ^{[1
]}

Gil, S ^{[1
]}

Mestres, R ^{[1
]}

Parra, M ^{[1
]}

机构：

[1] Univ Valencia, Dept Quim Organ, Valencia, Spain

来源：

SYNLETT | 1999年 / 07期

关键词：

pyridones; isoquinolones; lithium enolates; carboxylic acids;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

We report a simple procedure for the preparation of 4,6-disubstituted and 3,4,6-trisubstituted-2-pyridones and 3-substituted-1-isoquinolones, in good yields, from lithium dienediolates of alpha,beta-unsaturated carboxylic acids and nitriles.

引用

页码：1088 / 1090

页数：3

共 23 条

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