Regiospecific alkylation of histidine and histamine at C-2

被引：38

作者：

Jain, R ^{[1
]}

Cohen, LA ^{[1
]}

ElKadi, NA ^{[1
]}

King, MM ^{[1
]}

机构：

[1] GEORGE WASHINGTON UNIV,DEPT CHEM,WASHINGTON,DC 20052

来源：

TETRAHEDRON | 1997年 / 53卷 / 07期

关键词：

D O I：

10.1016/S0040-4020(96)01193-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The first regiospecific synthesis of 2-alkyl-L-histidines and 2-alkylhistamines starting from fully protected L-histidine and histamine via silver catalyzed radical decarboxylative oxidation of alkylcarboxylic acids by ammonium persulfate in 10% H2SO4 is described. (C) 1997, Elsevier Science Ltd.

引用

页码：2365 / 2370

页数：6

共 50 条

[1] Regiospecific alkylation of histidine and histamine at N-1 (c)
Tetrahedron, 15 (5363):
[2] Regiospecific alkylation of histidine and histamine at N-1 (tau)
Jain, R
Cohen, LA
TETRAHEDRON, 1996, 52 (15) : 5363 - 5370
[3] REGIOSPECIFIC ALKYLATION OF HISTIDINE AND HISTAMINE AT N-1 (TAU) AND ANTIMALARIAL ACTIVITIES OF THE ANALOGS
JAIN, R
COHEN, LA
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1995, 210 : 217 - MEDI
[4] THE REGIOSPECIFIC ALKYLATION OF HISTIDINE SIDE-CHAINS
JONES, JH
RATHBONE, DL
WYATT, PB
SYNTHESIS-STUTTGART, 1987, (12): : 1110 - 1113
[5] C-2/C-3 annulation and C-2 alkylation of indoles with 2-alkoxycyclopropanoate esters
Bajtos, Barbora
Yu, Ming
Zhao, Hongda
Pagenkopf, Brian L.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2007, 129 (31) : 9631 - 9634
[6] Regiospecific bromination of cephalosporin sulfones at C-2 with cyanogen bromide
Gunda, TE
Szoke, GN
SYNTHETIC COMMUNICATIONS, 1997, 27 (19) : 3395 - 3403
[7] HYDROGEN-DEUTERIUM EXCHANGE OF THE C-2 PROTONS OF HISTIDINE AND HISTIDINE PEPTIDES AND PROTEINS
BRADBURY, JH
CHAPMAN, BE
CROMPTON, MW
NORTON, RS
TEH, JS
JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 2, 1980, (04): : 693 - 699
[8] ASSIGNMENT OF C-2 HISTIDINE PROTON MAGNETIC RESONANCES OF RIBONUCLEASE-A
BRADBURY, JH
CHAPMAN, BE
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1972, 49 (04) : 891 - &
[9] DOUBLY EXCITED-STATES OF C-2, C-2(+), AND C-2(2)+
BRUNA, PJ
WRIGHT, JS
JOURNAL OF MOLECULAR STRUCTURE-THEOCHEM, 1991, 76 : 213 - 218
[10] ALKYLATION OF PHENOL WITH C-2 AND C-3 ALCOHOLS OVER IRON CATALYST
GRABOWSKA, H
WRZYSZCZ, J
RESEARCH ON CHEMICAL INTERMEDIATES, 1992, 17 (03) : 263 - 270

← 1 2 3 4 5 →