Synthesis of 4-(1,3-dioxo-2,3-dihydro-1H-2-indenyl) substituted 1-benzylpyrrole-3-carboxylates via a tandem four-component reaction

被引：5

作者：

Alizadeh, Abdolali ^{[1
]}

Mokhtari, Javad ^{[1
]}

机构：

[1] Tarbiat Modares Univ, Dept Chem, Tehran, Iran

来源：

COMPTES RENDUS CHIMIE | 2013年 / 16卷 / 02期

关键词：

Pyrroles; Ninhydrin; 1-Phenyl-2-(1,1,1-triphenyl-lambda(5)-phosphanylidene)-1-ethanone; Enaminone; Multicomponent reaction; ONE-POT; ROUTE;

D O I：

10.1016/j.crci.2012.10.003

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

An efficient approach for the preparation of functionalized 4-(1,3-dioxo-2,3-dihydro-1H-2-indenyl) substituted 1-benzylpyrrole-3-carboxylates is described. This four-component reaction between ninhydrin, 1-phenyl-2-(1,1,1-triphenyl-lambda(5)-phosphanylidene)-1-ethanone, primary amines and alkyl acetoacetate proceeds in MeOH under reflux condition in good to excellent yields. (C) 2012 Academie des sciences. Published by Elsevier Masson SAS. All rights reserved.

引用

收藏

页码：105 / 108

页数：4

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