Synthesis and preclinical evaluation of carbon-11 labelled P2X7 receptor antagonists as PET tracers of microglial activation

被引：0
|
作者：
Janssen, Bieneke [1 ]
Wilkinson, Shane M. [2 ]
Ory, Dieter [3 ]
Vugts, Danielle J. [1 ]
van den Hoek, Johan J. [1 ]
Schuit, Robert C. [1 ]
Beaino, Wissam [1 ]
Kooijman, Esther J. M. [1 ]
Chishty, Mansoor [4 ]
van der Perren, Anke [5 ]
Baekelandt, Veerle [5 ]
Molenaar, Ger T. [1 ,6 ]
Funke, Uta [1 ,6 ]
Shevchenko, Rostislav V. [4 ]
Lammertsma, Adriaan A. [1 ]
Bormans, Guy [3 ]
Kassiou, Michael [2 ]
Windhorst, Albert D. [1 ]
机构：
[1] Vrije Univ Amsterdam Med Ctr, Radiol & Nucl Med, Amsterdam, Netherlands
[2] Univ Sydney, Sch Chem, Sydney, NSW, Australia
[3] Katholieke Univ Leuven, Lab Radiopharm, Dept Pharmaceut & Pharmacol Sci, Leuven, Belgium
[4] Pharmidex Pharmaceut Serv Ltd, London, England
[5] Katholieke Univ Leuven, Neurobiol & Gene Therapy, Dept Neurosci, Leuven, Belgium
[6] BV Cyclotron VU, Amsterdam, Netherlands
来源：
JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 2017年 / 60卷
关键词：
D O I：
暂无
中图分类号：
Q5 [生物化学];
学科分类号：
071010 ; 081704 ;
摘要：
O 034
引用
收藏
页码：S53 / S53
页数：1
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