Recent advance of the application of interrupted Fischer indolization toward bioactive indoline alkaloids

被引：33

作者：

Mo, Yuanzhao ^{[1
]}

Zhao, Jipeng ^{[1
]}

Chen, Weiping ^{[1
]}

Wang, Qiaofeng ^{[1
]}

机构：

[1] Fourth Mil Med Univ, Sch Pharm, Xian 710032, Shaanxi, Peoples R China

来源：

RESEARCH ON CHEMICAL INTERMEDIATES | 2015年 / 41卷 / 08期

关键词：

Interrupted Fischer indolization; Furoindolines; Pyrrolidinoindolines; Alkaloid; KOPSIA-FLAVIDA BLUME; C3-QUATERNARY INDOLENINES; CASCADE DEAROMATIZATION; NATURAL-PRODUCTS; IN-VITRO; (+/-)-ASPIDOPHYLLINE; AKUAMMILINE; TRYPTOPHOLS; INHIBITORS;

D O I：

10.1007/s11164-014-1707-5

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

The interrupted Fischer indolization is an efficient way to construct fused indoline ring systems present in a variety of natural alkaloids. This paper will review the application of this reaction towards furoindolines and pyrrolidinoindolines with bioactivity.

引用

页码：5869 / 5877

页数：9

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