Mild and efficient one-pot three-component synthesis of benzopyrimidoquinoline-tetraone derivatives in ionic liquids

被引：10
作者：
Du, Bai-Xiang [1 ]
Zhao, Bo [1 ]
Cai, Gan [1 ]
Li, Yu-Ling [1 ]
Wang, Xiang-Shan [1 ]
机构：
[1] Xuzhou Normal Univ, Sch Chem & Chem Engn, Jiangsu Key Lab Green Synthet Chem Funct Mat, Xuzhou 221116, Jiangsu, Peoples R China
来源：
JOURNAL OF CHEMICAL RESEARCH | 2012年 / 08期
基金：
中国国家自然科学基金;
关键词：
multicomponent reactions; ionic liquid; pyrimidoquinoline; MULTICOMPONENT REACTIONS; CHEMISTRY; CATALYSIS;
D O I：
10.3184/174751912X13384724679874
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
An efficient one-pot synthesis of 5-aryl-5,12-dihydrobenzo[g]pyrimido[4,5-b]quinoline-2,4,6,11(1H,3H)-tetraone derivatives via three-component reaction of aromatic aldehydes, 2-hydroxy-1,4-naphthoquinone and 6-aminouracil in ionic liquid [bmim]BF4 is reported. This method had the advantages of easier work-up, environmentally benign procedure, high yields and ease of recovery and reuse of reaction media.
引用
收藏
页码：453 / 456
页数：4
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