Solid-phase synthesis of apicidin A and a cyclic tetrapeptoid analogue

被引:13
|
作者
Berst, F
Ladlow, M
Holmes, AB
机构
[1] GSK Cambridge Technol Ctr, Cambridge CB2 1EW, England
[2] Univ Cambridge, Dept Chem, Cambridge CB2 1EW, England
关键词
D O I
10.1039/b110068h
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
The solid-phase synthesis of the antiprotozoal cyclic tetrapeptide apicidin A is reported and its synthetic accessibility is contrasted with that of a structurally similar reduced cyclic tetrapeptoid analogue.
引用
收藏
页码:508 / 509
页数:2
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