Synthesis of (S)-(-)-1,4-Diaryl-6-methyl-4-trifluoromethyl-3,4-dihydropyrimidine-2(1H)-thiones

被引：0

作者：

Golovach, N. M. ^{[1
]}

Sukach, V. A. ^{[1
]}

Vovk, M. V. ^{[1
]}

机构：

[1] Natl Acad Sci Ukraine, Inst Organ Chem, UA-02660 Kiev, Ukraine

来源：

RUSSIAN JOURNAL OF ORGANIC CHEMISTRY | 2012年 / 48卷 / 03期

关键词：

ANALGESIC ACTIVITY EVALUATION; PYRIMIDINE;

D O I：

10.1134/S1070428012030165

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

(S)-(+)-4-Amino-4-aryl-5,5,5-trifluoropentan-2-one reacted with aryl isothiocyanates containing electron-withdrawing substituents to give (S)-(-)-1,4-diaryl-6-methyl-4-trifluoromethyl-3,4-dihydropyrimidine-2(1H)-thiones.

引用

页码：430 / 433

页数：4

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